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N4-(1H-imidazol-2-ylmethyl)-N4-methyl-6-(propan-2-yloxy)pyrimidine-2,4-diamine
N-(2-methoxyethyl)-6-methyl-N-[(4-methylphenyl)methyl]pyridine-2-carboxamide
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4-methylphenyl)propan-1-one
3-[(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}pyrrolidin-3-yl)methyl]benzamide
2-{2-[2-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
5-(methoxymethyl)-N-(4-{5-methyl-4-[(4-methylpentanamido)methyl]-1,3-oxazol-2-yl}phenyl)furan-2-carboxamide
ethyl 1-(3-phenylprop-2-ynoyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
4-hydroxy-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}amine
6-[3-(pyrrolidine-1-carbonyl)phenyl]quinazolin-4-amine
1-(2-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)piperidin-2-one
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzene-1-sulfonamide
5-methanesulfonyl-1'-(6-methoxypyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(2,4,6-trimethylphenoxy)ethyl]thiolan-3-amine
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)prop-2-ene-1-sulfonamide
(4aS,8aR)-6-(1-methyl-1H-indole-6-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(2E)-3-(3-fluorophenyl)-1-{4-[2-(oxolan-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}prop-2-en-1-one
4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1-(2-phenylethyl)piperazin-2-one
4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5,6-dimethylpyrimidine
N-[(2-methoxyphenyl)methyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
dimethyl(3-{2-[1-(6-methylquinolin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
2-methoxy-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-(3-methylbutyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
(2S,4R)-4-amino-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-N-methylpyrrolidine-2-carboxamide
8-(cyclohex-3-en-1-ylmethyl)-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,9S)-11-({4-[(thiophen-2-ylmethyl)amino]quinazolin-2-yl}methyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
(3S,4R)-1-(3-carboxybenzoyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
2-[(4-methoxyphenyl)methyl]-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
[(3R,5S)-5-(morpholin-4-ylmethyl)-1-(3-phenylpropyl)piperidin-3-yl]methanol
1-(benzenesulfonyl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazine
N-(2,3-dihydro-1H-inden-2-yl)-N-propylquinoxaline-6-carboxamide
4-{6-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
(4S,4aS,8aS)-4-phenyl-1-(1,2,5-thiadiazole-3-carbonyl)-decahydroquinolin-4-ol
4-(pyridin-3-yl)-1-{[4-(thiolan-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-4-ol
(2R,3R,6R)-3-(4-fluorophenyl)-5-(2-propyl-1,3-thiazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperidin-3-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-[(2-fluoroethyl)sulfamoyl]benzamide
4-{1-[(3,4-difluorophenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
6-[(diethylamino)methyl]-N-[2-(1H-imidazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
6-[3-(dimethylamino)pyrrolidin-1-yl]-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(ethanesulfonyl)piperidine
N-({7-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-fluorobenzamide
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-methyl-1-[3-(1H-pyrazol-1-yl)phenyl]urea
2-(1-methyl-1H-1,2,3,4-tetrazol-5-yl)-N,N-bis(propan-2-yl)benzamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}propanamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-ol
ethyl 4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate