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1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-3-{2-[2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
{4-[(2,3-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-3-yl)methanol
1-ethyl-2-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-imidazole
1-({2-[(benzenesulfonyl)methyl]phenyl}methyl)-4-cyclopropyl-4-methylpyrrolidin-2-one
2-propyl-1-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazole
1-[(4-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)methyl]piperazine
N-methyl-1-(1H-pyrazol-1-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)cyclopropane-1-carboxamide
N-[(2R,3R)-2-methoxy-1'-(2-phenoxyacetyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
(2S,4R)-4-amino-N-ethyl-1-(3-methylfuran-2-carbonyl)pyrrolidine-2-carboxamide
3-acetyl-N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1H-pyrazole-5-carboxamide
1-[(4,5-dimethylfuran-2-yl)methyl]-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
methyl 5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-5-oxopentanoate
2-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N-methylacetamide
N,N,5-trimethyl-2-[3-(piperidin-1-yl)azetidin-1-yl]pyrimidin-4-amine
2-[(3,4-dimethoxyphenyl)methyl]-6-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
methyl 4-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]piperazine-1-carboxylate
N4-methyl-N2-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-2,4-diamine
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
5-chloro-2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
2-{3-[(1-methylpiperidin-4-yl)methyl]-5-[(oxan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
2-{2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
(2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(1,3-thiazol-2-ylmethyl)pyrrolidine-2-carboxamide
(3aS,6aR)-3-[2-(pyridin-2-yl)ethyl]-5-(pyridin-4-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-2-(2-methyl-1H-imidazol-1-yl)acetamide
N-ethyl-1-oxo-N-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(4aS,7aR)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(5-{[(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
2-methyl-1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}pentane-1,4-dione
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-(1-methyl-2-oxopyrrolidin-3-yl)benzene-1-sulfonamide
(3S)-1-(1-benzoxepine-4-carbonyl)-N,N-dimethylazepan-3-amine
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]thian-4-amine
N,N-dimethyl-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}azepan-4-amine
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
2-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-4-carbonitrile
5-[(4-chlorophenyl)methyl]-5-{3-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-[(1-{6-[(oxolan-3-ylmethyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(2R)-2-amino-N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}propanamide
methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
4-(3-ethoxy-4-methoxyphenyl)-1-(1H-imidazol-2-ylmethyl)-1H-1,2,3-triazole
4-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-1-(2-methoxyethyl)piperidine
2-(ethylsulfanyl)-5-[(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)methyl]pyrimidine
6-[2-(3-methoxyphenoxy)ethyl]-2,3-dihydro-1H-indol-2-one
N-methyl-5-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(3-chloro-2-fluorophenyl)-1-[3-(3-oxopiperazin-1-yl)propyl]urea
N-[(2,6-difluoro-3-methylphenyl)methyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}benzamide
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-3-(5-methylfuran-2-yl)benzamide
N-[(2,4-difluorophenyl)methyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-cyclohexyl-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-[(3-chloro-2-fluorophenyl)methyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one