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3-[5-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
N-[2-(naphthalen-1-yl)ethyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(piperidin-1-yl)ethyl]amine
2-(2-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[1-(3,4-dimethoxybenzoyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-(4-methoxyphenyl)-1-[2-(methylsulfanyl)benzoyl]piperidin-3-amine
3-(3-fluorophenyl)-4-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperazin-2-one
(1R,3S)-7-(4-chloro-2-fluorobenzoyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
ethyl 1-(4,4,4-trifluorobutan-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methylpropanamide
(5S,9aS,9bS)-5-(6-methoxy-2H-chromen-3-yl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(4aS,7aR)-1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3,4-dihydro-2H-1-benzopyran-3-yl)-3-[2-(piperidin-1-ylmethyl)phenyl]urea
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-[1-(naphthalen-1-yl)ethyl]acetamide
N-(2-methoxyethyl)-N-methyl-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
1-[2-(dimethylamino)-4-{[3-(1H-1,2,4-triazol-1-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(1-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-2-yl)methanol
1-methyl-N-(2-methylpropyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclopropyl-5-[2-(4-fluorophenyl)acetyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
2-chloro-4-[1-({2-[(dimethylamino)methyl]phenyl}methyl)-1H-imidazol-2-yl]phenol
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-(dimethylamino)-2-(4-methylphenyl)acetamide
ethyl({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
N-(1-{7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
4-[(2-chloro-4-fluorophenyl)methyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
1-(6-methoxy-4-methylquinazolin-2-yl)-N-(3-phenylpropyl)pyrrolidine-2-carboxamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
1-cyclohexanecarbonyl-N-(4H-1,2,4-triazol-4-yl)pyrrolidine-2-carboxamide
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-[(1-ethylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(2-methyl-1-benzofuran-5-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
3-(2-methyl-1-benzofuran-7-yl)-1-[1-(pyrazin-2-yl)piperidin-3-yl]urea
2-[(4-{5-[(cyclohexylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenol
2-{[2-amino-6-(isoquinolin-5-yl)pyrimidin-4-yl]amino}ethan-1-ol
N-(1-{7-[(2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
N4-[cyclopropyl(3-methylpyridin-2-yl)methyl]-5-ethyl-6-methylpyrimidine-2,4-diamine
2-(2-ethyl-1H-imidazol-1-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
(3aS,6aS)-2-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carbonitrile
[(3R,4R)-1-[(4-chloro-3-fluorophenyl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-{[7-(pyrimidin-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}pent-4-enamide
2-{2-methoxy-5-[(3-propylmorpholin-4-yl)methyl]phenoxy}acetic acid
1-(2-methylpropyl)-8-(pyridin-2-ylmethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(4-chlorophenyl)methyl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
2-(8-methoxyquinolin-5-yl)benzene-1-sulfonamide
5-cyclopropyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1,3-oxazole-4-carboxamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-(3-methylthiophene-2-carbonyl)piperidine