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2-cyclohexyl-1-(2-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-7-yl)ethan-1-one
N-(adamantan-1-yl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
methyl 4-(methylsulfanyl)-2-({5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazol-3-yl}formamido)butanoate
5-(4-methyl-1H-pyrazol-1-yl)-2-(4H-1,2,4-triazol-4-yl)pyridine
1-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(4-fluorophenyl)-4-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-1,4-diazepane
N-cyclopropyl-4-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}piperazine-2-carboxamide
3-[3-(dimethylamino)propyl]-5-[(2-methylphenyl)methyl]-5-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
(2S,4S)-4-amino-1-(4-aminopyridine-2-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4,6-dimethyl-2-oxo-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1,2-dihydropyridine-3-carboxamide
5-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
N-[(3-hydroxypyrrolidin-3-yl)methyl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
3-(2-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
1-{4-[(1-methoxybutan-2-yl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
10-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
methyl 2-{[5-(4-fluorophenyl)-4-{1-[(2E)-4-methylpent-2-enoyl]piperidin-3-yl}pyrimidin-2-yl]sulfanyl}acetate
2-cyclopropyl-5-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]pyrimidine
1-[3-(4-methylphenoxymethyl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
4-(1-methyl-1H-pyrazol-4-yl)-6-(piperidin-1-yl)pyrimidine
(2S,4R)-4-amino-N-(propan-2-yl)-1-[3-(thiophen-3-yl)propanoyl]pyrrolidine-2-carboxamide
{1-[(2-fluoro-5-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
2-cyclopentyl-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-(1,3-benzothiazol-2-yl)-3-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}propanamide
1-(4-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-4-methoxyphenoxy}piperidin-1-yl)ethan-1-one
3-(2-oxo-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)imidazolidine-2,4-dione
(3R,4R)-1-[2-(2-chloro-4-methylphenoxy)ethyl]-4-(hydroxymethyl)piperidin-3-ol
N-[(1R,3R)-3-aminocyclopentyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-(3-{4-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
(1S,5R)-6-(5-ethyl-1,3-oxazole-4-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-(3-fluorophenyl)-8-methoxy-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
3-[2-(3,4-difluorophenyl)ethyl]-1-(1-methylcyclopropanecarbonyl)piperidine
methyl 3-[(4-fluoro-3-methoxyphenyl)methyl]-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-cyclopropyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)-4-phenylbenzamide
1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1-methylpiperidin-4-yl)pyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethylpyrimidine-5-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
2-[(2,6-dimethylphenyl)amino]-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]propanamide
N-cyclopropyl-3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propanamide
3-[1-(3-methylphenyl)-1H-1,3-benzodiazol-2-yl]propan-1-ol
4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-(1-{7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
3-(azocan-1-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
4-(2-phenylpyrrolidine-1-carbonyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
N-(1,2-oxazol-3-ylmethyl)-2-(thiophen-2-yl)acetamide
5-{1-[2-(3,5-difluorophenyl)acetyl]piperidin-4-yl}-5-methyl-3-(pyridin-4-ylmethyl)imidazolidine-2,4-dione
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-[2-(2-fluorophenoxy)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
1-ethyl-N-{[1-(4-fluorophenyl)cyclopentyl]methyl}-5-oxopyrrolidine-3-carboxamide