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1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-(2-methoxyphenyl)ethan-1-one
N-(2-methyl-1-benzofuran-5-yl)-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-[(3S,4R)-1-(1H-indole-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
4-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-2,6-dimethylphenyl acetate
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-(1H-indol-1-yl)ethan-1-one
3-(2-{6-[(3-fluorophenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepan-1-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
9-(5-propylpyrimidin-4-yl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
3-phenyl-4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrazole
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-[3-(3-fluorophenyl)phenyl]-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-4-carboxamide
2-{4-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
N-(4-fluoro-2-methylphenyl)-3-[1-(furan-3-carbonyl)piperidin-3-yl]propanamide
5-(4-chlorophenyl)-3-[3-(methoxymethyl)piperidin-1-yl]-1,2,4-triazine
N-[(2-chloro-6-fluorophenyl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[(2,3-difluorophenyl)methyl]-5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)amine
methyl 4-({3-[1-(2-methylpropanamido)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)benzoate
4-(5-{[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]methyl}-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl)-2-methylpyridine
2-(adamantan-1-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3-methyl-1-phenylpiperazin-2-one
{1-[3-(azepane-1-carbonyl)-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperidin-4-yl}methanol
(3S,4R)-4-(3-fluorophenyl)-1-[(3-hydroxyphenyl)methyl]pyrrolidine-3-carboxylic acid
(1R,2S)-1-[(6-methyl-2-propylpyrimidin-4-yl)amino]-2,3-dihydro-1H-inden-2-ol
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)-4-sulfamoylbenzamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-ethenyl-N-methylbenzamide
N-butyl-N-methyl-3-({[(1R,2S)-2-phenylcyclohexyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
7-(cyclopropylmethyl)-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
ethyl 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-{[(1-methoxypropan-2-yl)amino]methyl}-1H-pyrazole-4-carboxylate
2-[4-(1-benzothiophene-5-carbonyl)morpholin-3-yl]acetic acid
ethyl 4-[4-(3-methyl-1-phenyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxylate
2-[(3,4-difluorophenyl)methyl]-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(1S,6R)-3-methyl-9-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
methyl 5-[(1-ethylpiperidin-4-yl)amino]-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-[(diethylamino)methyl]-N-(2,3-dihydro-1H-inden-2-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl 3-(oxolane-3-amido)-1-(2-phenylethyl)-5-[(quinolin-5-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-[2-(1,4-dimethylpiperazin-2-yl)acetyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(morpholin-4-yl)ethyl]-5-(thiomorpholine-4-carbonyl)piperidin-2-one
5-chloro-2-(2-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrrol-1-yl)pyridine
2-methyl-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(pyrrolidin-1-yl)propan-1-one
1-[4-(2-phenyl-1H-imidazol-1-yl)phenyl]ethan-1-ol
2-{3-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]phenoxy}ethan-1-ol
N-[(3S,4R)-1-(3-ethoxypropanoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
methyl 3-[(3-hydroxy-4-methoxyphenyl)methyl]-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-benzyl-N-(2-phenoxyethyl)-1,3-benzoxazole-5-carboxamide
N,2-dibenzyl-3-oxopiperazine-1-sulfonamide
5-acetyl-N-[1-(2-phenylethyl)piperidin-3-yl]thiophene-3-carboxamide
6-(cyclopentylamino)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide