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N-[1-(6-methylpyridin-3-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
3-(4-fluorophenyl)-N-(1,2-oxazol-5-ylmethyl)-3-phenylpropanamide
(3R,4S)-4-cyclopropyl-1-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}pyrrolidin-3-amine
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylbutanamide
2-cyclopropyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4-methylpyrimidine
N,N-dimethyl-2-{[2-(oxan-2-ylmethoxy)acetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
6-[1-(3-methoxyphenoxy)ethyl]-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
5-(5-ethyl-2-methylpyrimidin-4-yl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-(2-{[ethyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)ethan-1-one
N-[(3-phenoxyphenyl)methyl]-2-(pyrrolidin-3-yl)acetamide
3-(3-fluorophenyl)-N-methyl-N-[3-(oxolan-2-yl)propyl]-1H-pyrazole-4-carboxamide
1-[4-(4-{[(3-methylphenyl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
5-(piperidin-1-yl)-2-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-2,3-dihydropyridazin-3-one
1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
4-ethyl-3-({1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[4-(4-{[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
1-[(2-fluorophenyl)methyl]-N-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]propanamide
N-[2-(3-methoxyphenyl)-1-[1-(3-methyl-2-oxopentanoyl)piperidin-4-yl]ethyl]-N,3-dimethylbutanamide
4,6,7-trimethyl-2-{4-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-1-yl}quinazoline
(2S,4S)-N-ethyl-4-(5-methylthiophene-3-amido)-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1H-pyrazol-4-yl)propanamide
4-(1-acetylpiperidine-4-carbonyl)-6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(trifluoromethoxy)benzene-1-sulfonamide
4-(1H-imidazol-2-yl)-1-(4-methyl-5-phenylthiophene-2-carbonyl)piperidine
N-{3-[methyl(phenyl)amino]propyl}-2-propyl-1,3-thiazole-4-carboxamide
N-[(3R,4S)-1-(2-methoxyethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]cyclobutanecarboxamide
3-(4-chlorophenyl)-1-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]piperidine
1-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}cyclobutane-1-carboxamide
1-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
5-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
4-(pyrrolidine-1-carbonyl)-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidine
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-hydroxy-3-[({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)amino)methyl]-1-[(3-methoxyphenyl)methyl]piperidin-2-one
1-(2-methyl-4-{[3-(pyridin-3-yloxy)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
7-[(3-methylphenyl)methyl]-2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.5]decane
1-[(2-hydroxy-6-methoxyphenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
3-[2-(dimethylsulfamoyl)ethyl]-1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
3-butyl-4-ethyl-1-{2-[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-(2-hydroxy-3-methoxypropyl)-N-methylpyridin-2-amine
N,N,3,6-tetramethyl-2-(2-methylpyrimidin-5-yl)quinoline-4-carboxamide
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1,3-thiazol-4-ylmethyl)piperidine
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
methyl 6-[2-({2-[3-(trifluoromethyl)phenyl]acetamido}methyl)-2,3-dihydro-1-benzofuran-7-yl]pyridine-3-carboxylate
7-(2-methoxyacetamido)-1-methyl-2-phenyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,3-benzodiazole-5-carboxamide
7-fluoro-N,3-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1-benzofuran-2-carboxamide
(1R,2S)-2-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}cyclopentane-1-carboxamide
4-{1-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]ethyl}phenol