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(1R,3S)-7-(3-hydroxynaphthalene-2-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-{4-[(cyclopropylamino)methyl]-2-methoxyphenoxy}-3-(diethylamino)propan-2-ol
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-{5-methylthieno[2,3-d]pyrimidin-4-yl}piperazine
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
(4S)-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
4-(4-chlorophenoxy)-1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperidine
2-ethoxy-5-(2-{[(2S)-oxolan-2-ylmethyl]amino}pyrimidin-4-yl)benzoic acid
7-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
1-(3-methanesulfonamidophenyl)-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
N-(2,5-dimethylphenyl)-N'-(2-hydroxy-3-phenylpropyl)propanediamide
N-ethyl-2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}pyridine-4-carboxamide
3-[4-(3-chlorophenoxy)piperidin-1-yl]-5-(4-fluorophenyl)-1,2,4-triazine
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-2-ylsulfanyl)acetamide
N,N-dimethyl-6-(3-{1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrimidin-4-amine
1-[2-(dimethylamino)ethyl]-4-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one
2-{[(6-chloropyridin-3-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
6-ethyl-2-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}quinoline-4-carboxamide
2-{4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
8-(3,4-dimethoxybenzoyl)-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
(2E)-N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-3-(4-methoxyphenyl)prop-2-enamide
2-(2-{[cycloheptyl(methyl)amino]methyl}phenyl)-6-ethyl-3,4-dihydropyrimidin-4-one
N-cyclopropyl-4-[({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)amino]pyridine-2-carboxamide
N-(5-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-2-methylphenyl)butanamide
5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
methyl 3-[(3S,4R)-1-{[4-(diethylamino)phenyl]methyl}-4-(dimethylamino)piperidin-3-yl]propanoate
N-butyl-3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[(4-fluorophenyl)methyl]-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]propanamide
4-(4-chlorophenyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]butanamide
3-[2-(3,5-difluorophenyl)acetyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2S,4S)-N-ethyl-1-(naphthalen-1-ylmethyl)-4-[(pyridin-4-ylmethyl)amino]pyrrolidine-2-carboxamide
(1R,7S)-3-(2-ethoxyethyl)-N-methyl-4-oxo-N-(pyrimidin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N,2,6-trimethyl-N-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
6-(piperidin-1-yl)-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]pyrimidin-4-amine
1-(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-ol
N-(1-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide
N-[1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-2-(3-methoxyphenyl)ethyl]-N-methylfuran-2-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
(1S,5R)-3-(3-methoxy-2,2-dimethylpropanoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]acetamide
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl})amine
1-[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]-1,4-diazepan-5-one
2-(4-{[2-(5-methylfuran-2-yl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
2-(ethylamino)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}pyrimidine-5-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
N-[(3S,4R)-1-{[3-(furan-2-yl)phenyl]methyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-[(E)-2-phenylethenyl]pyridine-3-carbonitrile