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(2R)-2-amino-3-methyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
1-cyclopentyl-N-[2-(4-methoxyphenyl)propan-2-yl]-6-oxopiperidine-3-carboxamide
(3S,9R)-N-benzyl-2,8-dioxo-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-11-carboxamide
8-[2-(1H-indol-3-yl)acetyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
2-butyl-4-(1-methyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-ethoxy-6-{[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
6-[(4-fluorophenyl)methoxy]-4-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}-1-(propan-2-yl)-1,4-diazepan-2-one
N-cyclopropyl-4-{[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)sulfamoyl}benzamide
2-({2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)acetamide
({5-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[(2-methoxyphenyl)methyl]benzamide
1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-3-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
2-[2-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]-N-(pyridin-4-ylmethyl)acetamide
5-amino-N-(4-methoxy-3-pentanamidophenyl)-1H-pyrazole-3-carboxamide
[(3-methoxyphenyl)methyl](methyl){[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(pyrazin-2-yl)propanamide
(2S,3S)-2-{[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]formamido}-3-methylpentanamide
N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}oxolane-2-carboxamide
methyl 1-{[4-(3,3-dimethylbutanoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)propanamide
(1-methyl-4-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperazin-2-yl)methanol
N-(2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}ethyl)pyridine-3-carboxamide
7-(2,3-dimethoxyphenyl)-4-[(4-ethylphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(5-methylpyrazin-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-chloro-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(4-{[4-(1-benzofuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
6-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-9H-purine
dimethyl[(5-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}thiophen-3-yl)methyl]amine
N-({2-[3-(2,5-dimethylfuran-3-amido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-methyl-1H-indole-2-carboxamide
methyl 1-benzyl-3-cyclopropaneamido-5-{[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
5-methyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
3-ethyl-5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazole
2-methyl-4-(4-{1-[3-(1H-1,2,4-triazol-1-yl)phenyl]-1H-imidazol-2-yl}phenyl)but-3-yn-2-ol
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[3-(4-phenylbenzoyl)piperidin-1-yl]ethan-1-one
2-cyclopropyl-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[1-(methoxymethyl)cyclopentyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
4-{1-[2-(2-oxopiperidin-1-yl)acetyl]piperidin-3-yl}benzoic acid
1-[1-(4-methoxybenzenesulfonyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-tert-butyl-2-cyclobutyl-1-methyl-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
N-{1-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]-2-phenylethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
1-(adamantan-1-yl)-4-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
N-[2-(methylsulfanyl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
5-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methylacetamide
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-methyl-N-[1-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]butanamide
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide