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[(3-{[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-benzyl-N-butyl-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
1-(1-cyclopropylethyl)-5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H,4H-pyrazolo[3,4-d]imidazole
methyl (2S)-1-[1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]pyrrolidine-2-carboxylate
2-(1H-1,3-benzodiazol-1-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethan-1-one
5-[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-methyl-5-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-pyrazole
N3-cyclooctyl-N5-(furan-2-ylmethyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-[4-(5-ethyl-2-methylpyrimidin-4-yl)phenoxy]acetic acid
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[methyl({[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl})amino]methyl}-4H-chromen-4-one
4-[2-(3,4-dichlorophenyl)morpholin-4-yl]-4-oxobutane-1-sulfonamide
3-ethyl-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
N-[2-(2-ethylpyrimidine-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
(2S,4R)-4-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-N-ethyl-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
1-(furan-2-ylmethyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]piperidine-4-carboxamide
1-cyclopropyl-3-(4-methoxyphenyl)-3-{2-oxo-2-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
3-(3,4-difluorobenzoyl)-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-{[3-(3,5-dimethylphenyl)propanamido]methyl}-N-methylfuran-2-carboxamide
2-[3-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-(piperidin-1-yl)pyridine
1-(3-{[7-(5-chloropyridin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1H-indol-1-yl)ethan-1-one
N'-({1-[(2,5-dimethylphenyl)methyl]piperidin-3-yl}methyl)ethanediamide
N-(2H-1,3-benzodioxol-5-yl)-3-[4-(methylsulfanyl)benzoyl]piperidine-1-carboxamide
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(ethyl)methylamine
2-[(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amino]-N-[2-methyl-6-(propan-2-yl)phenyl]acetamide
N5-(2-methoxyethyl)-N6-(2,2,2-trifluoroethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(furan-2-yl)pyrimidine
2-cyclobutyl-1-methyl-N-[2-(4-methylphenyl)ethyl]-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
6-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-9H-purine
4-[2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-[(3R,4R)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
N-[(3,4-difluorophenyl)methyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
2-[1-cyclohexyl-4-(5-phenyl-1,2,4-oxadiazol-3-yl)piperazin-2-yl]ethan-1-ol
N-{1-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)(oxolan-2-ylmethyl)amine
6-(pyrrolidin-1-ylmethyl)-4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1,4-oxazepan-6-ol
4-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
4-(4-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)phenol
[(1-cyclopentylpiperidin-4-yl)methyl][(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl](oxolan-2-ylmethyl)amine
4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
ethyl({[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}){[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-(but-2-yn-1-yl)-5-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
5-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-5-[(2-chlorophenyl)methyl]imidazolidine-2,4-dione
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-ol
4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
2-amino-6-(2-amino-5-methyl-1,3-thiazol-4-yl)-4-(5-ethylfuran-2-yl)pyridine-3-carbonitrile
2-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N-methylacetamide