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6-methyl-1-(3-oxo-3-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}propyl)-1,2-dihydropyridin-2-one
(3S,4R)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
[(3R,4R)-1-(1-benzothiophen-2-ylmethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-(7-methoxy-4-methylquinazolin-2-yl)-N-methyl-N-(oxan-2-ylmethyl)piperidin-4-amine
3-chloro-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
2-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-3,4,7-trimethyl-1H-indole
5-methoxy-2-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-1,3-benzodiazole
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2-methoxyphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-[4-(2-chlorobenzoyl)piperazin-1-yl]-2-[(3-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-methyl-1-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[(2-methylbutyl)sulfamoyl]benzamide
methyl 3-acetamido-5-{[4-(4-methoxyphenyl)butan-2-yl]amino}-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
9-[2-(morpholin-2-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-6-methylpyridine-2-carboxamide
(1-{[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}benzoic acid
{9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-methyl-1-[(4-phenylphenyl)methyl]pyrrolidine-2-carboxamide
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-2-methylfuran-3-carboxamide
5-[(4-methoxyphenyl)methyl]-1-methyl-N-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl (2S)-2-{[2-(dimethylamino)-2,3-dihydro-1H-inden-2-yl]formamido}-2-phenylacetate
2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)-N-{[8-(2-phenylacetyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-3-methoxypropanamide
4-(1H-pyrazol-1-yl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylic acid
1-[7-(3-methylfuran-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-3-ol
[(3-ethoxy-4-methoxyphenyl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
1-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
4-benzyl-3-[1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidine-1-carboxamide
9-[(2R)-2-amino-3-methoxypropanoyl]-2-cyclobutyl-2,9-diazaspiro[5.5]undecan-3-one
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-[(prop-2-en-1-yl)amino]benzamide
(1S,5R)-6-(2-ethoxybenzoyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(3-ethyladamantan-1-yl)-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[3-(4-methylphenoxymethyl)piperidin-1-yl]propan-1-one
2-[9-(4-methylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
{1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethylpiperidin-3-yl}methanol
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-3-(1H-imidazol-4-ylmethyl)piperazin-2-one
ethyl 2-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carboxylate
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dimethyl-1H-indole-7-carboxamide
3-(4-methoxyphenyl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-pyrazole-5-carboxamide
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxylate
1-(2-oxo-2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)pyrrolidin-2-one
2-(3-fluorophenyl)-N-[4-(4-{[2-(3-methoxyphenyl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
5-(3-hydroxy-3-phenylpyrrolidine-1-carbonyl)-2-(3-methylphenyl)pyrimidin-4-ol
2-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]pyridin-3-ol
(1R,3S)-3-(2-aminoethoxy)-7-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol