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N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-7-fluoro-2-methylquinoline-4-carboxamide
3-(4-fluoro-3-methylphenyl)-1-methyl-6-(2-phenylethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
ethyl 4-benzyl-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxylate
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}-1-(2-methylpropyl)piperidine
2-(6-methoxypyridin-3-yl)-1,3-benzoxazole
5-[(dimethylsulfamoyl)amino]-N-[(3-fluorophenyl)methyl]-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-(3-aminobenzoyl)-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
3-[({1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-{[1-(phenoxymethyl)cyclopropyl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
2-chloro-4-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}phenol
2-[2-(benzyloxy)ethyl]-N,N-dimethylbenzamide
2-ethyl-7-(2-methoxybenzamido)-N,1-dimethyl-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
5-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
2,4-difluoro-N-(oxolan-2-ylmethyl)-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,4-diazepan-2-one
5-(dimethylamino)-2-[2-(morpholin-4-yl)ethyl]-2,3-dihydropyridazin-3-one
3-(4-phenylbenzoyl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-(1-cyclopentyl-4-hydroxypiperidin-4-yl)-1-benzofuran-2-carboxamide
3-(2-methylpropyl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1,2-oxazole-5-carboxamide
4-{2-[1-(1,3-thiazol-4-ylmethyl)piperidin-2-yl]ethyl}morpholine
6-[(3-ethoxy-4-methoxyphenyl)methyl]-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
7-chloro-4-hydroxy-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylquinoline-3-carboxamide
1-{4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-2-(3,4,5-trimethoxyphenyl)ethan-1-one
N-[3-(1,3-benzothiazol-2-yl)propyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-[(2-chlorophenyl)methyl]-5-[1-(4-ethenylbenzoyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
7-(cyclopropylmethyl)-2-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-(5-ethyl-1,3,4-thiadiazol-2-yl)propanamide
4-[1-(4-methoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-3-methyl-1-propyl-1H-pyrazole
4-(4H-1,2,4-triazol-4-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]benzamide
ethyl 1-(but-3-enoyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
N-[(2R,3R)-1'-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
N-{[1-(2-methyl-1,3-benzothiazol-6-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
methyl 4-[5-(furan-3-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]benzoate
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
7-(2-methoxyethyl)-2-{pyrazolo[1,5-a]pyridine-3-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
2-methoxy-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
3-[1-(4,4,4-trifluorobutyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(1-methyl-1H-indazol-6-yl)piperazine-1-carboxamide
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
(1-{2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-4-yl)(pyridin-2-yl)methanol
N-[(3R,4R)-3-hydroxy-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidin-4-yl]pyrazine-2-carboxamide
5-[1-(2-methoxyacetyl)piperidin-4-yl]-5-(2-methylpropyl)-3-(thiophen-2-ylmethyl)imidazolidine-2,4-dione
(1R,6S)-3-({2-[4-(1H-imidazol-1-yl)butoxy]phenyl}methyl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane
N-[(3-methoxyphenyl)methyl]-N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-(3-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}phenyl)ethan-1-amine
2-(methylsulfanyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,3-thiazole-4-carboxamide