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8-[4-(dimethylamino)pyrimidin-2-yl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-(1-methyl-1H-imidazol-2-yl)-3-(1-phenylcyclopropyl)-1,2,4-oxadiazole
{[5-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
methyl 1-(2-methoxyethyl)-5-{[(4-methoxyphenyl)methyl]amino}-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl 5-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(3-chloro-4-methoxyphenyl)-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
N-{[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
(1S,5R)-6-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-benzyl-1-{2-[3-(3,4-dimethoxyphenyl)propanamido]ethyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[2-(2-fluorophenyl)-2-hydroxyethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(2,2-dimethyloxan-4-yl)-1H-imidazole
2-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}-1-(pyridin-3-yl)ethan-1-ol
3-(4-fluoro-3-methylphenyl)-6-(4-methyl-1H-imidazole-2-carbonyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]azetidin-3-yl}-1H-pyrazole
2-(azepan-1-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
8-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(thiophen-3-yl)pyridine-3-carboxamide
5-cyclopropanecarbonyl-1'-(1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(2-methylpyridin-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
{2-[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}urea
dimethyl[1-(3-{1-[2-(pyridin-2-yl)ethyl]-1H-imidazol-2-yl}phenyl)ethyl]amine
6-{3-[benzyl(methyl)amino]piperidin-1-yl}pyridine-3-carbonitrile
9-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-4-(morpholin-4-yl)benzamide
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl][(2-methylphenyl)methyl](2-methylpropyl)amine
3-(1-methyl-1H-1,3-benzodiazol-5-yl)-1-[3-(4-methylpiperazin-1-yl)propyl]urea
1-methyl-5-(naphthalen-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
8-fluoro-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}quinoline-2-carboxamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-1-methylazepane-2-carboxamide
N-(2-methoxyethyl)-5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
ethyl 5-({[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}carbamoyl)-1H-imidazole-4-carboxylate
6-chloro-2-{2-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
N-(5-chloro-2-methoxyphenyl)-3-[1-(3,6-dimethylpyrazin-2-yl)piperidin-3-yl]propanamide
2-(furan-3-amido)-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-ylmethyl)piperidine
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-{1-[4-(piperidin-1-yl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
8-[(2-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(5-methylpyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[2-(benzyloxy)ethyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
methyl 3-({4-[2-(morpholin-4-yl)ethyl]piperazine-1-carbonyl}amino)benzoate
4-[2-(benzyloxy)benzoyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(1-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-2-one
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2,2-dimethyloxane-4-carboxamide
ethyl 5-[4-(furan-2-yl)benzoyl]-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(pyridin-3-ylmethyl)-4-[(4-{[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(2,5-dimethoxyphenyl)acetamide
5-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
5-[1-(3-cyclopentylpropanoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione