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(2E)-N-cyclopentyl-3-(3-fluorophenyl)-N-({4-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)prop-2-enamide
5-(2,6-difluorophenoxymethyl)-N-methyl-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide
(3R,4R)-3,4-dimethyl-1-[3-(morpholin-4-yl)benzoyl]pyrrolidin-3-ol
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-(2-phenylpropyl)-6-azaspiro[2.5]octane
2-(3-hydroxypropyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-cyclohexyl-5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-(oxan-4-yl)-1H-1,2,4-triazole
(2R)-2-amino-1-[3-(2-fluorophenoxy)azetidin-1-yl]-4-methylpentan-1-one
1-[1-(4-chlorophenyl)ethyl]-3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]urea
1-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3-fluorophenyl)methyl]piperidine-3,5-dicarboxamide
1-(furan-2-ylmethyl)-N-[3-(pyridin-2-yl)propyl]piperidine-3-carboxamide
1-(5-methoxy-2-methylphenyl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
methyl 5-(quinolin-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
6-hydroxy-2,5,7,8-tetramethyl-N-[3-(pyridin-3-yl)propyl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
N-cyclohexyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-({4-[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[methyl({[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl})amino]methyl}phenol
2-(1H-1,2,4-triazol-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]benzamide
2-[(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]-6-methylpyridine-3-carbonitrile
7-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
4-methyl-N-{2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propyl}benzamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
1-(cyclohex-3-en-1-ylmethyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-methyl-6-propyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-2-(1-ethylpiperidin-4-yl)ethan-1-one
5-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
N,2,2,6,6-pentamethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-amine
(4aS,7aR)-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[6-(4-ethylpiperazin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}[(3-fluorophenyl)methyl]amine
5-(2-propyl-1H-imidazol-1-yl)pyrazin-2-amine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-methyl-1-(oxan-2-ylmethyl)urea
2-(6-chloropyridin-3-yl)-1-[2-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
4-[5-(3-chloro-2-fluorobenzoyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
N-methyl-2-(morpholin-4-yl)-N-[(4-phenoxyphenyl)methyl]propanamide
ethyl 3-benzyl-1-[(2,6-dimethylphenyl)carbamoyl]piperidine-3-carboxylate
N-benzyl-N-(4-hydroxybutyl)-1,3,7-trimethyl-1H-indole-2-carboxamide
1-(3-methylbutyl)-3-(propan-2-yl)-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
1-tert-butyl-2-methyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
6-(2,2-dimethylpropyl)-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
3-{[8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenol
methyl 3-[(1-methyl-1H-indol-3-yl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)morpholine-4-carboxamide
1-(1-benzoxepine-4-carbonyl)-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
methyl 3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-5-{[(2-methylphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-(2-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one