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N-benzyl-5-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}pyrimidin-2-amine
1'-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-(pyridin-3-ylmethyl)propanamide
6-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-{2-[cyclohexyl(methyl)amino]ethyl}-8-(pent-4-enoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-methoxyethyl)-1-methyl-N-(pyridin-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[(5-methylfuran-2-yl)methyl]-3-propylpiperidine-3-carboxylic acid
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
2,5-dimethyl-3-{4-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}pyrazine
1-cyclopentyl-4-(2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazin-2-one
1-[cyclohexyl(methyl)amino]-3-[3-({[2-(4-fluorophenyl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-methoxy-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-3-{2-[4-(4-methylphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
(3S,7S)-5-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
(4aR,8aS)-1-(2,2-diphenylethyl)-6-(1H-indol-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
1-propyl-5-(4-propylpiperazin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-[(2-fluorophenyl)methyl]-3-(2-oxo-2-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}ethyl)piperazin-2-one
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-[4-(thiophene-2-carbonyl)piperazin-1-yl]propan-1-one
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-4-carbonitrile
5-[1-(2-acetylbenzoyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-acetamidoethyl)-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
[(2-butyl-1H-imidazol-4-yl)methyl](methyl)(quinolin-5-ylmethyl)amine
4-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,3-thiazole
(5S,9aS,9bS)-5-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-(benzyloxy)-1-cyclohexyl-4-(2,6-dimethylpyrimidine-4-carbonyl)-1,4-diazepan-2-one
(3aS,6aR)-5-(isoquinolin-5-ylmethyl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
ethyl 4-{1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}piperidine-1-carboxylate
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethylpiperidine-2-carboxamide
N-methyl-2-[3-({[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)carbamoyl}amino)phenyl]acetamide
N-(3-chloro-4-methylphenyl)-3-(4-ethoxypiperidin-1-yl)propanamide
2-ethyl-9-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]-4-propylpyrrolidine-3-carboxylic acid
N-ethyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(oxan-4-ylmethyl)propanamide
N-(2-{7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methylbenzamide
4-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
4-methyl-2-{2-oxo-2-[3-(pyrimidin-4-yl)piperidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
N-[(3R,4S)-1-[(2-aminopyrimidin-5-yl)methyl]-4-cyclopropylpyrrolidin-3-yl]-4,4,4-trifluorobutanamide
methyl (2S,4R)-1-[(2,4-dimethylphenyl)methyl]-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
N-[(2R,3R)-1'-(3-ethynylbenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
methyl 2-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
N-[4-(3-fluorophenyl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-ethyl-3-(3-fluorophenyl)-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-1H-pyrazole-4-carboxamide
2-cyclobutyl-5-fluoro-1-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-ethyl-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)pyrrolidine-2-carboxamide
8-[(4-chlorophenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(5-tert-butyl-1H-pyrazol-3-yl)-5,6,7-trimethoxy-1,2,3,4-tetrahydroquinolin-2-one