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N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-(propan-2-yl)piperidine-4-carboxamide
9-[(dimethyl-1,3-thiazol-5-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N3-ethyl-N1-[2-(pyridin-2-ylmethoxy)phenyl]pyrrolidine-1,3-dicarboxamide
2-(isoquinolin-5-ylmethyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
5-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2,1,3-benzoxadiazole
1-(cyclohexylmethyl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-amine
N-[2-(dimethylamino)ethyl]-1-{1-[2-(trifluoromethyl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
5-{2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-fluoro-N-(furan-2-ylmethyl)-N-methyl-4-oxo-1,4-dihydroquinoline-2-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(2,3,4,5-tetrafluorophenyl)methyl]acetamide
3-[(3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}phenyl)formamido]propanamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-(dimethylamino)-2,3-dihydro-1H-indene-2-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(diethylamino)ethyl]-1H-pyrazole-4-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidine-2-carboxamide
2-{4-[(4-methylphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
2-{4-[6,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
N-(2-{1-[(4-chloro-2-fluorophenyl)methyl]piperidin-2-yl}ethyl)acetamide
7-(2-methylphenyl)-9-(oxolan-3-yloxy)-4-(1H-pyrrol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[5-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
ethyl 4-{[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]carbamoyl}piperazine-1-carboxylate
N-[(3R,4R)-3-hydroxy-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]pyrazine-2-carboxamide
6-(2-fluoro-4-methoxyphenyl)-7-methyl-2-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-[(2-fluorophenyl)methyl]-N-{[3-(trifluoromethoxy)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-{1-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-1H-imidazol-2-yl}phenol
(4aS,7aR)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3,5-difluoro-4-(trifluoromethyl)phenyl]-3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
2-{4-[(5-ethylfuran-2-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
6-{2-[3-(dimethylamino)propyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carboxylic acid
5-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-2-[(phenylsulfanyl)methyl]pyrimidin-4-ol
3-(4-{[2-(2-phenylethynyl)phenyl]methyl}piperazin-1-yl)propanamide
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea
3-(1H-1,3-benzodiazol-2-yl)-1-(3-propylmorpholin-4-yl)propan-1-one
2-[4-(1H-imidazol-2-ylmethyl)piperazin-1-yl]-1,3-benzoxazole
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-(propan-2-yl)benzamide
N-[(2R,3R)-2-methoxy-1'-{[4-(pyrrolidin-1-yl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
(1S,6R)-3-methyl-9-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
[1-({1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
3-cyclohexyl-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1H-pyrazole-4-carboxamide
2-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-4,6-dimethylpyridine-3-carbonitrile
4-(3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
4-[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-[(4-methylphenyl)methyl]pyrrolidin-2-one
6-[3-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-2-cyclopropyl-1,3-benzoxazole
N-methyl-2-(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)acetamide
1-(4-methylpiperazin-1-yl)-3-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)propan-1-one
2-(1-ethyl-1H-pyrazol-4-yl)-4-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}quinoline
N-cyclohexyl-3-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
2-(2-methyl-1H-1,3-benzodiazol-5-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
(2R,3R)-3-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-methyl-3-(thiophen-3-ylmethyl)-5-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione