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N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(2-oxopyrrolidin-1-yl)acetamide
9-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-fluoro-N-methyl-2-oxo-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-methoxy-4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
[1-(4-methoxyphenyl)ethyl](methyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine
[2-(3,4-dimethoxyphenyl)ethyl](methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]propan-1-one
1-[(2-fluorophenyl)methoxy]-8-(2,3,4-trimethoxybenzoyl)-1,8-diazaspiro[4.5]decan-2-one
1-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-[2-(butan-2-yl)phenoxy]acetamide
2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-1-(pyridin-2-yl)ethan-1-ol
[3-({1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
dimethyl(3-{2-[1-(4-methylphthalazin-1-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
3-(5-fluoro-2-methoxybenzoyl)-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
(2S)-2-amino-N-ethyl-3-(1H-imidazol-4-yl)-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
1-(4-fluorophenyl)-3-(oxan-4-yl)-5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,4-triazole
N-[(2-methoxyphenyl)methyl]-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(3R,4S)-1-{[4-(4-chlorophenyl)phenyl]methyl}-4-(dimethylamino)piperidin-3-yl]propan-1-ol
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
5-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
2,4-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
(1R,3S)-7-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-7-azaspiro[3.5]nonane-1,3-diol
4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-N,N-dimethylpiperazine-1-sulfonamide
3-(3-acetylphenyl)-1-(3-methylbut-2-en-1-yl)-6-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-({cyclopropyl[(3-methylthiophen-2-yl)methyl]amino}methyl)benzene-1,2-diol
1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}azepan-4-ol
1-(2,3-dimethylphenyl)-4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
(3R)-N-[2-(2-fluorophenoxy)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(1-benzyl-1H-1,2,4-triazol-5-yl)-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
2-({[1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-1,3,4-thiadiazole
[(1-methyl-1H-imidazol-2-yl)methyl][(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amine
(1S,5R)-6-propyl-3-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 4-benzyl-1-[3-(methylsulfanyl)propyl]piperidine-4-carboxylate
methyl 1-benzyl-3-cyclopropaneamido-5-[(4-hydroxy-4-methylpentan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]acetamide
N-[(2,3-dimethoxyphenyl)methyl]-1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperazine-1-sulfonamide
{4-[({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]phenyl}methanol
9-[2-(ethylamino)pyrimidine-5-carbonyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
3-hydroxy-3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(2-phenylethyl)piperidine
1-ethyl-3-(2-methylphenyl)-3-[2-oxo-2-(4-propylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
5-(2-methylpropyl)-1'-(5-propylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]propan-1-one
2-[4-(5-methyl-4-phenyl-1H-imidazol-1-yl)butyl]pyridine
2-(benzyloxy)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
4-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]-3-(4-fluorophenyl)piperazin-2-one