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3-(3-methylpiperidin-1-yl)-1-(4-phenylpiperazin-1-yl)propan-1-one
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
N-(1-{2-oxo-2-[4-(quinazolin-2-yl)piperazin-1-yl]ethyl}-1H-pyrazol-4-yl)thiophene-3-carboxamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-acetyl-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
4-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
1-cyclopentyl-3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
(2E)-N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-3-(4-methoxyphenyl)prop-2-enamide
2-(2,2-dimethyloxan-4-yl)-4-{3-[4-(2-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-(1H-pyrazol-1-yl)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]butan-1-one
N-{[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-(2-ethyl-6-methylphenyl)-4-[5-(pyridin-3-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
6-methyl-3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1,2-dihydropyridin-2-one
N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
5-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2-methoxyphenol
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(4-methoxyphenyl)furan-2-carboxamide
2-(3-hydroxypropyl)-8-(5-methylthiophene-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-N-methylbenzamide
1-[2-({1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidin-4-yl}amino)ethyl]cyclopentan-1-ol
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylthiophene-2-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1,2-oxazole-5-carboxamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
(4aR,7aS)-1-benzyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-1-(3-phenoxybenzoyl)piperazine-2-carboxamide
2-(4-methoxyphenyl)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
N-(1-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
N-methyl-3-{[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
1-(ethanesulfonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
4-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-4-(2-oxopyrrolidin-1-yl)butanamide
(2S,4R)-1-[(3-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N,N-dimethylpyrrolidine-2-carboxamide
2-(5-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-(4-methyl-1,3-oxazole-5-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(1H-indol-1-yl)ethyl]-N-methylacetamide
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidine
[(1-methyl-1H-pyrazol-4-yl)methyl]({6-methyl-2-[(2-methylphenyl)methoxy]quinolin-3-yl}methyl)amine
7-chloro-2-methyl-4-(1-methylpiperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(azepane-1-sulfonyl)-5-(quinolin-8-yl)benzoic acid
N-methyl-1-(4-methylquinazolin-2-yl)-N-(oxan-2-ylmethyl)piperidine-4-carboxamide
1-(2-methylpyridin-4-yl)-4-(1,3-thiazol-4-ylmethyl)-1,4-diazepane
4-(3-{[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amino}propanamido)benzamide
3-[ethyl({[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl})amino]-1λ6-thiolane-1,1-dione
N-ethyl-N-[2-(2-methylphenoxy)ethyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
(3S,5S)-5-(4-methylpiperazine-1-carbonyl)-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
2-{1-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]pyrrolidin-3-yl}benzoic acid
5-methyl-1-(3-methylbutyl)-4-phenyl-1H-imidazole
N4-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-methylpyrimidine-2,4-diamine
methyl 6-(cyclohex-3-ene-1-carbonyl)-2-[(3,5-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate