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5-(6-methyl-2-phenyl-1,2-diazinane-1-carbonyl)-2-(pyridin-3-yl)pyrimidin-4-ol
(3R,4R)-4-(hydroxymethyl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-ol
1-methyl-4-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}piperazine
(3S,5R)-N3-(4-methylphenyl)-N5-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3,5-dicarboxamide
1-benzyl-5-acetamido-2-methyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1H-1,3-benzodiazole-7-carboxamide
1-(benzyloxy)-8-(3-cyclopentylpropanoyl)-1,8-diazaspiro[4.5]decan-2-one
7-methoxy-4-methyl-2-{4-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}quinazoline
(3aS,6aR)-3-cyclopentyl-5-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 3-(5-methyl-1,2-oxazole-3-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(2-chloro-4-fluorophenoxymethyl)-N,N-dipropyl-1,2-oxazole-3-carboxamide
3-[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]-4,5,6,7-tetrahydro-2H-indazole
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyrazin-2-yl)propan-2-yl]pyridin-2-amine
1,4,6-trimethyl-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
9-[(1S,3R)-3-aminocyclopentanecarbonyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(thiolan-3-yl)pyrimidin-2-amine
(1S,5R)-6-benzyl-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
7-fluoro-3-{[methyl(thiophen-3-ylmethyl)amino]methyl}-1-[2-(phenylsulfanyl)ethyl]-1,2-dihydroquinolin-2-one
(4aR,8aS)-6-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
(3R,4R)-1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}-4-(morpholin-4-yl)piperidin-3-ol
5-[6-amino-5-cyano-4-(1-ethyl-5-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
3-{[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl]amino}-2,2-dimethylpropan-1-ol
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[(2-methylphenyl)methyl]amino}piperidin-1-yl)phenyl]acetamide
1-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
1-[(3-{[1-(4-fluorobenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
4-fluoro-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
(1S,5R)-6-benzyl-3-[2-(benzyloxy)ethyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(2,6-difluorophenyl)methyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
3-(cyclohex-3-en-1-ylmethyl)-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-[2-(1H-imidazol-2-yl)benzoyl]-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-ethyl-2-[1-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1H-imidazol-2-yl]-1H-1,3-benzodiazole
1-(2-ethoxyethyl)-N,N-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-methyl-7-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}-1,2-dihydroquinolin-2-one
7-(cyclopropylmethyl)-N-(4-ethylphenyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
8-[(2,4-dimethylphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)-1,3-thiazole-5-carboxamide
1-[2-({[3-(3-fluorophenyl)oxolan-3-yl]methyl}amino)ethyl]imidazolidin-2-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclopent-3-ene-1-carboxamide
8-(6-cyclopropylpyrimidin-4-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
{1-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}methanol
2-cyclopropanecarbonyl-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
5-[2-(2-methoxyphenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}pyrimidine-5-carboxylic acid
2-(4-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
(3S,5R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
3-{1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropanoyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one