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6-{[2-(methylcarbamoyl)piperidin-1-yl]methyl}pyridine-2-carboxylic acid
4-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,2-dimethylpiperazine
N-[(2,5-dimethoxyphenyl)methyl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanamide
5-butyl-1-(2-methoxyphenyl)-4-(1-methyl-1H-pyrrole-2-carbonyl)piperazin-2-one
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
1-[(6-chloro-4-oxo-4H-chromen-3-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(4-chlorophenoxy)-1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
4-[(2-chlorophenyl)methyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-5-one
N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(quinolin-5-ylmethyl)acetamide
1-(4-chloro-2-methoxy-5-methylphenyl)-3-[2-(diethylamino)ethyl]-3-methylurea
1-(1H-imidazol-4-ylmethyl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylic acid
2-chloro-N-(1-{1-[(2-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
methyl 4-({[(3S,5S)-5-(methylcarbamoyl)-1-(naphthalen-1-ylmethyl)pyrrolidin-3-yl]amino}methyl)benzoate
3-cyclohexyl-N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
9-methoxy-7-(5-methylthiophen-2-yl)-4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{2-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-8-methylquinolin-3-yl}methanol
N-[(2R,3R)-1'-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-4-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}benzamide
5-(azepan-1-yl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
3-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamido]-N-phenylpropanamide
1-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)azepane
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(4,4,4-trifluorobutyl)piperidin-4-ol
N-({7-[(2,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrazolo[1,5-a]pyridine-7-carboxamide
1-(dimethyl-1,3-oxazole-5-carbonyl)-N-(furan-2-ylmethyl)piperidine-4-carboxamide
N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-(3-hydroxypropyl)-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amino}pyrimidin-4-yl)piperidin-4-ol
N-(2-methoxy-5-methylphenyl)-7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepine-2-carboxamide
4-(1H-pyrazol-3-yl)-N-{3-[(pyridin-3-yl)amino]propyl}benzamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)propanamide
N-(1-benzothiophen-5-ylmethyl)-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
(3aR,6aR)-2-(dimethylcarbamoyl)-5-(5-propyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[({3-[4-(furan-3-yl)-6-oxo-1,6-dihydropyrimidin-2-yl]phenyl}methyl)(methyl)amino]-N,N-dimethylacetamide
N-butyl-3-({[(4-ethylphenyl)methyl](methyl)amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
4-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazole-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
2-amino-6-butanoyl-4-(3-fluorophenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-cycloheptyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[(2R,3R)-1'-(2,1,3-benzothiadiazol-5-ylmethyl)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2-cyclopropylpyrimidine
2-(2H-1,3-benzodioxol-5-yl)-8-methoxy-5-(3-methylbut-2-en-1-yl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
(1S,2S,9S)-11-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
5-cyclopropyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,3-oxazole
7-[2-(1H-pyrazol-1-yl)butanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-(3,4-difluorophenoxymethyl)-3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazole