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1-cyclobutanecarbonyl-N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-fluorophenyl)methyl]piperazin-2-one
4-methyl-N-{3-[2-(pyridin-3-yl)-1H-imidazol-1-yl]propyl}benzene-1-sulfonamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(6-methylpyridine-3-carbonyl)piperidine-4-carboxamide
N-[(2R,3R)-2-hydroxy-1'-(thiophen-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
N-(1-methyl-1H-1,2,3-triazol-4-yl)-2-[4-methyl-3-(1-methyl-1H-pyrazol-5-yl)-1H-pyrazol-1-yl]acetamide
2-{[4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]amino}-1-(1-methyl-1H-imidazol-2-yl)ethan-1-ol
2-methyl-N-[3-(5-methyl-4-{[2-(2-methylphenyl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]furan-3-carboxamide
(3R,4R)-1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
3-(5-methyl-1H-pyrazol-1-yl)-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)propanamide
1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
N-[1-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)piperidin-4-yl]methanesulfonamide
7-[(2-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-4-yl}-6-(pyrrolidin-1-yl)pyrimidine
(1R,5S,8S)-3-{[5-(3-chlorophenyl)furan-2-yl]methyl}-3-azabicyclo[3.2.1]octan-8-ol
2-{[2-(4,5-dimethylfuran-2-yl)-1H-imidazol-1-yl]methyl}pyridine
(pyridin-4-ylmethyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
7-(cyclobutylmethyl)-2-[(4-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[4-({1-[1-(2-methylpentyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)piperazin-1-yl]ethan-1-one
1-[(4,8-dimethoxynaphthalen-1-yl)methyl]-3-(hydroxymethyl)pyrrolidin-3-ol
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)propanamide
(3R,4R)-4-ethyl-1-(6-phenylpyridine-2-carbonyl)piperidine-3,4-diol
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[2-(1H-indol-3-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
2-ethyl-1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}butan-1-one
N-(cyclobutylmethyl)-3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(oxolan-2-ylmethyl)propanamide
2-(2-{[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
5-{[1-(2,5-dimethylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-1,3,4-thiadiazol-2-amine
(3R,4R)-4-(azepan-1-yl)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-ol
2-{4-[(4-methoxy-3-methylphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-[(3S,4R)-1-(3-hydroxynaphthalene-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-[2-(dimethylsulfamoyl)ethyl]-2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-(2-fluorophenyl)-4-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
4-chloro-N,N-dimethyl-5-{1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}-1,3-thiazol-2-amine
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
5-({3-[3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
N-{3-hydroxy-4-[2-(trifluoromethyl)morpholine-4-carbonyl]phenyl}acetamide
4-(2-hydroxybenzoyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(6-oxo-1,6-dihydropyridine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[(3,5-dimethylphenyl)methyl]-4-[2-(ethylsulfanyl)propanoyl]piperazin-2-one
2-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-1,2-oxazolidin-4-ol
2-{4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1H-pyrazol-1-yl}-N-methylacetamide
2-(4-chlorophenyl)-4-[3-(1H-imidazol-2-yl)benzoyl]morpholine
4,6-dimethyl-2-oxo-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
3-[(3R,4S)-3-[5-(hydroxymethyl)furan-2-amido]-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
(1S,5R)-6-(cyclobutylmethyl)-N-methyl-7-oxo-N-phenyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-benzoyl-1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidine
N-(4-methoxyphenyl)-3-(3-phenylpropanoyl)piperidine-1-carboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
N-[(3-fluorophenyl)methyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide