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1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N,N-bis(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{[2-(aminomethyl)piperidin-1-yl]methyl}-6-methylquinolin-4-ol
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2,5-dimethoxybenzamide
4-[1-(5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-3-yl]benzoic acid
1-(2-methylpropyl)-N-[2-(pyridin-3-yl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(4-fluorophenoxymethyl)-1-{3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine
{1-[2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]piperidin-4-yl}methanol
6-(aminomethyl)-2-(2-{[4-(1,3,5-triazin-2-yl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1-(pyridin-2-yl)piperidine-3-carboxamide
4-[4-(piperazin-1-ylmethyl)phenoxy]thiane-4-carboxylic acid
2-(1-benzofuran-2-yl)-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}acetic acid
2-methoxy-4-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-3-carbonitrile
N-{2-[1-(2,3-dimethylphenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
[2-(2-amino-1,3-benzothiazol-5-yl)phenyl]methanol
(2R)-2-[(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propanamide
5-(1-ethyl-3-methyl-1H-pyrazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(1,3-benzothiazol-2-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine
3-[2-(2-ethoxyphenyl)ethyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
2-[(dimethylamino)methyl]-4-(pyridin-2-yl)phenol
4-chloro-N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzene-1-sulfonamide
2-(1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
1-(furan-2-ylmethyl)-4-[3-(1H-pyrazol-4-yl)benzoyl]piperazine
N-methyl-N-(2-phenoxyethyl)-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
5-methyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
4-(3-methylphenoxy)-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-(methylsulfanyl)benzamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
1-[1-(4-chloro-2-hydroxybenzoyl)piperidin-3-yl]pyrrolidin-2-one
(3S,4R)-N,N-dimethyl-4-propyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidin-3-amine
(4aR,7aS)-4-[(3-ethoxyphenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-(furan-2-carbonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-cyclopropyl-N-({4-methoxy-3-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-3-(2-methoxyphenyl)propanamide
1-[2-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-oxoethyl]-1,2-dihydropyrimidin-2-one
4-{pyrazolo[1,5-a]pyridine-3-carbonyl}morpholine-2-carboxylic acid
1-(cyclopropylmethyl)-N-methyl-5-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-3-ol
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[2-(propan-2-yloxy)ethyl]benzamide
8-(furan-2-ylmethyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]propanamide
3-ethyl-1-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]urea
8-[2-(methylamino)acetyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-[(2,3-difluorophenyl)methyl]-2-(3-methyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-(3-chlorophenyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-phenylpropanamide
1-[(3-methoxyphenyl)methyl]-N-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}piperidin-3-amine
({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)({[4-(methylsulfanyl)phenyl]methyl})propylamine
3-{1-[2-(3-methoxyphenoxy)ethyl]piperidin-3-yl}benzoic acid
3-({methyl[(3-phenyl-1H-pyrazol-5-yl)methyl]amino}methyl)pyrrolidin-3-ol
N1-{4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}pentane-1,5-diamine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(1H-pyrazol-1-yl)butanamide
2-fluoro-N-[3-(1H-imidazol-1-yl)propyl]-6-methoxy-N-(pyridin-4-ylmethyl)benzamide