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6-(2,3-dihydro-1-benzofuran-2-carbonyl)-3-(4-fluoro-3-methylphenyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-[(cyclohex-3-en-1-ylmethyl)amino]-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-5-(phenylsulfamoyl)benzamide
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]urea
5-(3,4-diethoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
6-(2-chlorophenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{1-[6-(2-aminoethyl)pyrimidin-4-yl]piperidin-4-yl}piperidin-4-ol
2-{[(3S,4S)-3-carboxy-4-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole-4-carboxylic acid
3-(3-hydroxyquinoxalin-2-yl)-1-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}propan-1-one
5-ethyl-3-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2-oxazole
N-butyl-N-[(2-fluorophenyl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
4-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-5-phenyl-2-(pyridin-3-yl)pyrimidine
2-(3-fluorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
2-[4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
3-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)imidazolidine-2,4-dione
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-4-(thiophen-2-yl)butan-1-one
2-methoxy-N-[1-(2-phenylethyl)-7-(pyrrolidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-8-fluoroquinoline-2-carboxamide
methyl (2S,4R)-4-(isoquinoline-5-amido)-1-methylpyrrolidine-2-carboxylate
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}propanamide
N-methyl-2-{4-[2-(thiophene-2-sulfonamido)acetyl]morpholin-3-yl}acetamide
1-{4-[(3-benzyl-1H-1,2,4-triazol-5-yl)methoxy]phenyl}-1H-1,2,3,4-tetrazole
2,3,5-trimethyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1-(3-methoxyphenyl)piperazin-2-one
2-ethyl-6-(4-methyl-5-phenylthiophene-2-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
2-acetyl-8-[2-(benzyloxy)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(1H-indol-3-yl)ethyl]acetamide
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)cyclopentane-1-carboxamide
5-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-4-amine
1-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-(3-methoxyphenyl)propan-1-one
1-{6-methyl-5-[5-(pyrazin-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}butan-1-one
N-(1-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N-ethyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(pentan-3-yl)acetamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-amine
2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(4-sulfamoylphenyl)methyl]acetamide
6-{[3-(dimethylamino)phenyl]methyl}-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
8-methoxy-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(1R,5S,6S)-3-{[3-(difluoromethoxy)phenyl]methyl}-N-(2-hydroxyethyl)-N-methyl-3-azabicyclo[3.1.0]hexane-6-carboxamide
1-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)-4-(4-fluorophenyl)butane-1,4-dione
6-methyl-1-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}propyl)-1,2-dihydropyridin-2-one
3-(3-fluorophenyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-1H-pyrazole-4-carboxamide
3-(3-fluoro-4-methoxybenzoyl)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
phenyl (7S,9aR)-7-[(4-chlorophenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
3-methyl-N-(1-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
4-(1H-imidazol-1-ylmethyl)-1-(1H-pyrazole-4-carbonyl)piperidine
1-[(3-methoxyphenyl)methyl]-4-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)piperazin-2-one
2-(3-methoxyphenoxymethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1,3-oxazole-4-carboxamide