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2-(3-fluorophenyl)-2-hydroxy-N-[2-(2-oxopyrrolidin-1-yl)ethyl]acetamide
2,2-diphenyl-1-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
N-(3-cyano-4-ethoxyphenyl)-4-(furan-3-carbonyl)-1,4-diazepane-1-carboxamide
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-{1-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]piperidin-4-yl}-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-[1-(2,3,6-trifluorobenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
3-({4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine
5-(2-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
5-hydroxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrazine-2-carboxamide
2-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-phenylacetamide
N-cyclobutyl-2-{4-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]morpholin-3-yl}acetamide
7-(3,6-dimethylpyrazin-2-yl)-4-(pyrimidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}propanoic acid
4-{2-[3-(propan-2-yloxy)phenyl]pyridine-4-carbonyl}morpholine
{4-benzyl-1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methanol
N'1-[2-(4-cyclohexylmorpholin-2-yl)ethyl]cyclopropane-1,1-dicarboxamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-[1-butyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
(3aR,6aS)-5-(2,3-dihydro-1H-indene-5-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-N-[2-(4-fluorophenyl)ethyl]-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
4-(1H-indol-2-ylmethyl)-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[4-(hydroxymethyl)phenyl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(quinolin-8-yloxy)ethyl]acetamide
1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-N-phenylpiperidin-3-amine
2-methoxy-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
methyl 3-(2-methoxyacetamido)-1-methyl-5-{[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[(4-methoxynaphthalen-1-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-cyclopropyl-1-[1-(6-cyclopropylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
N-(1-oxo-1-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pentan-2-yl)acetamide
1-ethyl-N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}piperidine-3-carboxamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(piperazin-1-yl)ethan-1-one
1-(4-chloro-3-fluorobenzoyl)-N-phenylpiperidin-3-amine
N-cyclopropyl-N-[2-phenyl-1-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]furan-2-carboxamide
3,3,3-trifluoro-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}propan-1-one
1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]urea
2-methyl-1-{4-[2-(oxolan-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
5-[(4-benzylpiperidin-1-yl)methyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(1-cyclopentyl-1H-imidazol-2-yl)benzonitrile
8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5-{1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
5-chloro-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,2-dimethylbenzamide
5-chloro-6-(2,3-dihydro-1-benzofuran-7-yl)-2-methylpyrimidin-4-ol
1-[1-(3-phenylpropyl)piperidin-4-yl]-N-[(3S)-pyrrolidin-3-yl]piperidine-4-carboxamide
1-[(2S,4R)-1-[(2,6-difluorophenyl)methyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
3-(3-fluoro-4-methoxybenzoyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
2-[(2,3-dimethoxyphenyl)methyl]-4-{4-[2-(3-methylphenyl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-methanesulfonyl-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-amine
4-{4-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine