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N-[(3,4-dimethoxyphenyl)methyl]-2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
(3S,4S)-1-(2-aminopyrimidin-4-yl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
N-(1-{1-[3-(2-chlorophenyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
methyl 6-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(dimethylamino)-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}butan-1-one
4-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3,3-dimethylpiperazin-2-one
1-benzyl-3-(pyridin-2-ylmethyl)-8-(quinolin-6-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(2-butoxyacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(adamantan-1-yl)-3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-benzyl-N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetamide
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-[3-(methylsulfanyl)propyl]-1H-1,3-benzodiazole-7-carboxamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(3-methylfuran-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-3-(thiophen-2-yl)propan-1-one
4-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-1,3-dimethyl-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid
3,5-dimethoxy-N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}urea
4-[2-(2-chlorophenyl)-2-hydroxyethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-methoxy-N-{1-methyl-5-[3-(2-methylphenyl)piperidine-1-carbonyl]-2-(pyridin-3-yl)-1H-1,3-benzodiazol-7-yl}acetamide
(1R,5R)-3-benzoyl-6-{[3-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
6-ethoxy-2-{4-[(2-methoxyphenyl)methyl]-1,4-diazepan-1-yl}-4-methylquinazoline
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-5-(methoxymethyl)furan-2-carboxamide
3-(azocane-1-sulfonyl)-N-(oxan-4-yl)benzamide
1-[2-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-3-ol
1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-5-(2,3,6-trifluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})amine
2-[(3-methoxyphenyl)amino]-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]butanamide
N-[2-(4-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}morpholin-2-yl)ethyl]acetamide
3-[2-(4-cyclohexylpiperazin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
(3aS,6aR)-5-(3-ethyl-1H-pyrazole-5-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
6-(4-ethylphenyl)-N,N-bis(prop-2-en-1-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
9-[(2R)-2-amino-3-methoxypropanoyl]-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
N-(adamantan-2-yl)-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
methyl(oxan-2-ylmethyl){[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-(2-fluoro-5-methylphenyl)-4-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-4-oxobutanamide
4-[2-(2-methoxyphenoxy)acetyl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-({7-fluoro-2-[4-(3-methoxyphenyl)piperazin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)furan-3-carboxamide
3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-[3-(1H-1,2,4-triazol-1-yl)propyl]benzamide
1-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-3-(oxolan-2-ylmethyl)urea
2-(2,5-dioxoimidazolidin-4-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(propan-2-yl)piperidine-3-carboxamide
(3aS,6aS)-5-(1-benzofuran-5-ylmethyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[(4-methoxyphenyl)methyl]carbamoyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
{2-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}urea
5,6-dimethyl-2-[3-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-3-(thiophen-2-yl)propan-1-one
4-methyl-1-(4-{5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidin-4-yl}piperidin-1-yl)pentan-1-one
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-3-(2-oxopyrrolidin-1-yl)benzamide
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-2-(trifluoromethyl)pyrimidin-4-amine