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dimethyl({[(1R,5S,6S)-3-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(2,4,5-trimethylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
1-[(2-chloro-4-fluorophenyl)methyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(5-methyl-4-{[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]-3-phenoxypropanamide
1-{2-[2-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
N-[2-(oxan-2-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
methyl 2-(tert-butylsulfamoyl)-6-[(4-methoxy-2,3-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
9-(2-chlorobenzoyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{5-[2-(diethylamino)ethyl]-1,3,4-thiadiazol-2-yl}-1-[2-(5-methylfuran-2-yl)ethyl]urea
3-[1-tert-butyl-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylpropanamide
1-(butane-1-sulfonyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
2-[2-(3-chloro-4-methoxyphenyl)phenyl]ethan-1-amine
2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
2-(2-chloro-6-fluorophenyl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
9-(4-ethenylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(3-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)methyl]morpholine
N-[2-(dimethylamino)ethyl]-2-fluoro-6-hydroxy-N-[(3-methylthiophen-2-yl)methyl]benzamide
1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-4-carboxamide
6-(4-methoxyphenyl)-9-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-6,9-diazaspiro[4.5]decan-7-one
1-(2-aminoethyl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
6-{[5-(furan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-methylpyrimidin-4-ol
3-(2-methylphenyl)-3-(2-oxo-2-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}ethyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
7,7-dimethyl-2-(1H-1,2,3,4-tetrazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-acetyl-N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}benzamide
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-2,6-dimethoxybenzamide
1-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
N'-cyclopropyl-N-(4-methylphenyl)-N'-(3-phenylprop-2-yn-1-yl)propanediamide
2-[(3R,4S)-3-(1-tert-butyl-1H-pyrrole-3-amido)-4-propylpyrrolidin-1-yl]acetic acid
3-methyl-1-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,2-dihydroquinoxalin-2-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(1H-1,2,3-benzotriazol-1-yl)propanamide
N-(cyclobutylmethyl)-2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-(oxolan-2-ylmethyl)acetamide
4-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazine-1-carboxamide
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-phenylbutanamide
4-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
6-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1,3-benzothiazole
1-[(2S,4R)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-[(4-ethoxyphenyl)methyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
2-[1-(5-chloro-2-methoxyphenyl)-5-(1-methyl-2-oxo-1,2-dihydropyridin-4-yl)-1H-1,2,4-triazol-3-yl]acetamide
3-[methyl({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl})amino]-N-(pyridin-3-yl)propanamide
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
1-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-4-phenylpiperidine-4-carbonitrile
4-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]-1λ6-thiane-1,1-dione
8-[4-(furan-2-yl)benzoyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
3,5-difluoro-N-{[8-(pyridine-2-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
N-[1-(2-phenylethyl)piperidin-3-yl]-2-(trifluoromethyl)benzamide
3-{2-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-(3-fluorobenzenesulfonyl)-3-[4-(methylsulfanyl)benzoyl]piperidine
{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}methanamine