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3-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-indole-2-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(1H-1,2,3-benzotriazol-4-yl)-1-(thiolan-3-yl)urea
2-{[(6-methoxypyrimidin-4-yl)amino]methyl}-3,4-dihydroquinazolin-4-one
2,6-dimethoxy-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}pyridine-3-carboxamide
1-(1,3-benzothiazol-2-yl)-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-amine
N-(2,3-dihydro-1H-inden-2-yl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(3R,4R)-4-ethyl-1-(5-phenyl-1,3-oxazole-4-carbonyl)piperidine-3,4-diol
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-[3-(pyridin-3-yl)phenyl]urea
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl][(3-methoxyphenyl)methyl](prop-2-en-1-yl)amine
methyl 7-oxo-3-(3-phenylpropanoyl)-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-benzyl-3-ethyl-1-[4-(1H-pyrazol-1-yl)butanoyl]-1,4-diazepan-5-one
7-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
8-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidine
1-[(2-chlorophenyl)methyl]-4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-ethyl-3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-{imidazo[1,2-a]pyridin-3-yl}acetamide
2-(methylsulfanyl)-4-{3-[1-(oxolan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
4-(benzyloxy)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine
(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]{[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-[1-(thiolan-3-yl)piperidin-4-yl]imidazolidine-2,4-dione
3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]propanamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(2-methylphenyl)-1H-indazol-1-yl]acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}morpholine
8-[(3,4-dimethoxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-fluorobenzamide
1-methyl-4-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-{[7-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-2-methoxy-N-[(3S)-2-oxoazepan-3-yl]acetamide
3-cyclopentaneamido-N-[(1-propyl-1H-pyrazol-4-yl)methyl]benzamide
(1R,9S)-5-amino-3-(5-chlorothiophen-2-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-methoxy-1-{1'-[2-(4-methylpiperidin-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-8-methyl-2,8-diazaspiro[5.5]undecane
4-(2-methoxyethyl)-3-({4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}methyl)-4H-1,2,4-triazole
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
3-(3,4-dimethyl-1H-pyrazol-5-yl)-1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[8-(propan-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
N-(2-{[5-(furan-3-yl)-4-(4-methylphenyl)pyrimidin-2-yl]amino}ethyl)acetamide
1-[3-(4-fluorophenyl)phenyl]-N-[2-(1H-pyrazol-1-yl)ethyl]piperidin-4-amine
N,5,7-trimethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
3-({1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
[1-(1,3-benzothiazol-2-ylmethyl)-4-benzylpiperidin-4-yl]methanol
2-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}-1-(2-methylpropyl)-1H-1,3-benzodiazole
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)ethane-1-sulfonamide
1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-methoxyethan-1-one
4-benzyl-3-{1-[(2S)-5-oxopyrrolidine-2-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
8-(5-methylpyrazine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one