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N-{[1-(naphthalen-2-ylmethyl)piperidin-4-yl]methyl}cyclopropanecarboxamide
2-amino-3-ethyl-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-butyl-1-(4-chlorophenyl)-4-(1H-pyrazole-3-carbonyl)piperazin-2-one
(7R,9aR)-7-(hydroxymethyl)-6,9-dioxo-N-phenyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-ethyl-N-(4-hydroxybutyl)quinoxaline-5-carboxamide
2-(dimethylamino)-N-[2-(4-fluorophenyl)-1-{1-[3-(trifluoromethyl)benzoyl]piperidin-4-yl}ethyl]-N-methylacetamide
N-[1-(1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-methylbutanamide
N-({1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
ethyl 4-benzyl-1-[(6-acetamidoquinolin-2-yl)methyl]piperidine-4-carboxylate
2-methoxy-2-phenyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-6-methoxyhexan-1-one
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-4-methyl-1,3-oxazole-5-carboxamide
1-cyclohexyl-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
4-[5-(oxolan-3-ylmethyl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]benzamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,2-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
[(3R,4R)-1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-cyclohexanecarbonyl-1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
{1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-yl}methanamine
1'-[1-(4,6-dimethylquinazolin-2-yl)piperidine-4-carbonyl]spiro[indene-1,4'-piperidine]
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)(pyridin-3-ylmethyl)amine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
15-methyl-13-oxo-N-[2-(pyridin-4-yl)ethyl]-9-(thiophen-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(furan-2-carbonyl)piperidin-3-yl]propanamide
(3-{[1-(5-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-({8-[(2,5-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
N-(propan-2-yl)-3-{[(1-propyl-1H-pyrazol-4-yl)methyl]sulfamoyl}benzamide
3-[2-({3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrrol-1-yl]pyridine
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[1-(piperidin-1-ylmethyl)cyclohexyl]urea
1-methyl-3-(2-methylpropyl)-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-(oxan-4-yl)piperazin-2-yl}ethan-1-ol
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(propan-2-yloxy)ethan-1-one
2-cyclopentyl-N-{[8-(4-fluorobenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
2-(4-{2-[(4-chlorophenyl)amino]acetamido}-3,5-dimethyl-1H-pyrazol-1-yl)acetic acid
ethyl 1-(2,5-dimethylfuran-3-carbonyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
3-[2-(4-methylpiperazin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
N3-ethyl-N1-[2-methyl-4-(methylcarbamoyl)phenyl]pyrrolidine-1,3-dicarboxamide
3-(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
N-[2-(3-methoxyphenyl)ethyl]-6-[4-(methylsulfanyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-(furan-3-ylmethyl)piperidin-4-amine
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[3-(thiophen-2-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-({[2-(pyrrolidin-1-yl)ethyl]sulfanyl}methyl)-1H-1,2,4-triazole
(3R,4R)-4-(azepan-1-yl)-1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]piperidin-3-ol
2-(3-methoxyphenoxymethyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
N-(2-{[2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-6-(4-fluorophenyl)pyridin-3-yl]formamido}ethyl)acetamide
2-(4-ethylpiperazin-1-yl)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}ethan-1-one
3-(3,4-dimethoxybenzoyl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidine
5-(2-cyclopentylacetamido)-N-[(2-methoxyphenyl)methyl]-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
1-(2,6-dimethylpyridin-4-yl)-4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine