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N-({1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-benzyl-N-ethylpropanamide
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-ethyl-N-(1-hydroxypropan-2-yl)-1-benzofuran-3-carboxamide
N-[(3R,4R)-1-(5-acetylpyridin-2-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
[(4-fluorophenyl)methyl][(2E)-3-(furan-2-yl)prop-2-en-1-yl](pyridin-4-ylmethyl)amine
5-chloro-2-(4-ethylpiperazine-1-carbonyl)-3-phenyl-1H-indole
3-{[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]sulfonyl}-N-[2-(methylamino)ethyl]benzamide
N-[(3R,4R)-1-[(cyclohexylcarbamoyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
(3S,4S)-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
N-[(2R,3R)-1'-(2,4-dimethylbenzoyl)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
dimethyl({[(1-{[2-(2-phenylethynyl)phenyl]methyl}piperidin-3-yl)methyl]sulfamoyl})amine
2,5-dioxo-6-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-{6-[3-(methoxymethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-(2-oxoazepan-3-yl)propanamide
N-{1-[1-(2-phenylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-(1H-imidazol-2-ylmethyl)-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(2-methoxyethyl)-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(3-phenylprop-2-yn-1-yl)acetamide
5-[(3-methoxyphenyl)methyl]-5-{3-[3-(3-methylphenoxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
5-(3,4-difluorophenoxymethyl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1,2-oxazole-3-carboxamide
methyl 3-[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoate
(1R,5R)-6-[(2-ethoxyphenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3,6,7-trimethyl-N-[2-(2-oxopiperidin-1-yl)ethyl]-1-benzofuran-2-carboxamide
N-{2-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2,4-dimethylbenzamide
6-cyclopentyl-1-methyl-N-[1-(pyridin-3-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{1-[2-(2-chloro-4-fluorophenyl)acetyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-(1-benzyl-5-{spiro[2.5]octane-1-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)piperazin-2-one
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-(2,2,2-trifluoroethyl)-1H-1,3-benzodiazole-7-carboxamide
2-methyl-3-{[3-(pentan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2H-indazole
8-(1-cyclobutylethyl)-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-{1-[(3-chlorophenyl)methanesulfonyl]piperidin-2-yl}ethyl)acetamide
4-{4-[4-(2-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-[(2-fluorophenyl)methyl]piperidin-3-yl)methanol
2-methoxy-N-[3-(4-{[(2-methylphenyl)methyl]amino}piperidin-1-yl)phenyl]benzamide
1-methyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]sulfonyl}-1,2-dimethyl-1H-imidazole
6-{4-[5-phenyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
N-cyclooctyl-4-oxo-5-(piperidine-1-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
2-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
2-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]pyrazine
({[1-(1-benzofuran-2-carbonyl)piperidin-3-yl]methyl}sulfamoyl)dimethylamine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide
7-{[3-(pyridine-3-carbonyl)piperidin-1-yl]methyl}-4-(thiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[(prop-2-en-1-yl)amino]benzamide
N-cyclopropyl-1-(2-{1-[3-(4-methoxyphenyl)propanoyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
5-(1-{[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
methyl 3-({[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)propanoate