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3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-N-[(3-chlorophenyl)methyl]propanamide
2-methyl-6-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-[4-(3-methylphenyl)phenyl]-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1,8-naphthyridine-2-carboxamide
7-[(3-methylphenyl)methyl]-2-(1-phenyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
8-[(4-methyl-2-oxo-2H-chromen-7-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(1H-1,3-benzodiazol-2-ylmethoxy)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
1-methyl-2-{1-[2-(methylsulfanyl)benzoyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-{1-[4-(4-methoxybutyl)piperazine-1-carbonyl]cyclopentyl}-4-methylaniline
7-(cyclopropylmethyl)-2-[2-(1H-indol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
6-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-(2-{1-[1-(6-ethoxy-4-methylquinazolin-2-yl)pyrrolidine-2-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
1'-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]
2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyridin-3-ol
5-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2-hydroxy-1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
1-(1H-imidazol-2-ylmethyl)-N-[3-(1H-indol-2-yl)phenyl]pyrrolidine-2-carboxamide
N-({7-[(3,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)propane-2-sulfonamide
7-chloro-2-[(4-cyclopentylpiperazin-1-yl)methyl]-N-(oxolan-2-ylmethyl)quinazolin-4-amine
(4aS,8aS)-2-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-decahydroisoquinolin-4a-ol
N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazole-4-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(dimethylamino)-6-methylpyrimidin-4-yl]piperidin-4-yl}propanamide
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)isoquinoline-1-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-{[4-(hydroxydiphenylmethyl)piperidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(3-methoxyphenyl)-N-(2-phenoxyethyl)-1H-pyrazole-5-carboxamide
N-[(2R,3R)-2-(benzyloxy)-1'-(1H-indazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
2-[ethyl(methyl)amino]-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-{4-[hydroxy(phenyl)methyl]piperidin-1-yl}propan-1-one
7-(propan-2-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-cyclohexyl-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}acetamide
2-[3-(2-methylpropyl)-5-{[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,4-triazol-1-yl]pyridine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(thiophen-3-yl)propan-2-yl]benzamide
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-(9H-fluoren-2-yl)urea
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
2,6-dimethyl-8-{[(4-phenyloxan-4-yl)methyl]amino}octan-2-ol
ethyl 4-{6-[(3,4-dimethoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
2-methyl-8-[(4-phenoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-{2-[1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)propanamide
1-methyl-5-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-amino-3-(2-phenylpyrimidin-5-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methylbutan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-1H-indole-3-carboxamide
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-6-(5-oxo-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-(4-fluorophenyl)-N,N-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-{1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl}pyrrolidin-2-one
4-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-N-methyl-4-oxobutanamide
{3-[(2,4-difluorophenyl)methyl]-1-(furan-3-carbonyl)piperidin-3-yl}methanol
4-[(benzyloxy)methyl]-1-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one