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1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(7S,9aR)-N-(3-fluorophenyl)-7-[(1R)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
4-chloro-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-3-(1H-pyrrol-1-yl)benzamide
4-[(3aS,6aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-octahydropyrrolo[2,3-c]pyrrol-5-yl]-6-methylpyrimidin-2-amine
2-[(dimethylcarbamoyl)amino]-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
N-(2-hydroxyethyl)-1-{1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-{2-[1-(2-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]ethyl}morpholine
4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}morpholine
N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
[3-(2-phenoxyethyl)piperidin-3-yl]methanol
2-tert-butyl-N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
7-({7-ethyl-2,7-diazaspiro[4.4]nonan-2-yl}methyl)-4-(2-phenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(1-hydroxycyclohexyl)methyl]-4-(4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
2,6-difluoro-4-methoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
N-(1-{7-[(2-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
N-(butan-2-yl)-N-[(2-fluorophenyl)methyl]-2-hydroxypyridine-3-carboxamide
[5-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)furan-2-yl]methanol
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
1-[2-(cyclohexylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[2-(4-fluorophenyl)ethyl]piperidine-4-carboxamide
8-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-N,N-dimethyl-4-{[2-(methylsulfanyl)phenyl]methyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(5-phenylpentanoyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[4-(benzyloxy)phenyl]methyl}-4-(pyrrolidin-3-yl)piperazine
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(pyrazin-2-yl)piperidin-4-yl]oxy}benzamide
4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine
N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-6-methylpyridine-3-carboxamide
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-3,5-dimethyl-1-benzofuran-2-carboxamide
5-benzyl-5-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
1-cyclopentyl-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
(2S,3S)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methylpentanamide
4-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}piperazin-2-one
2-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,2-oxazinane
3-{[2-(2,3-dihydro-1H-inden-1-yl)acetamido]methyl}-N,N-dimethylbenzamide
1-[(2-fluorophenyl)methyl]-7-methoxy-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
(4aS,7aR)-1-[2-(4-fluorophenoxy)ethyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclooctyl-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
5-(butan-2-yl)-1-(pentan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)propanamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3,5-dimethoxybenzamide
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]piperazine-1-carboxamide
5,6-dimethyl-2-{[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
N-methyl-2-(2,3,4-trimethoxyphenyl)-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1-{2-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4-phenylpyrrolidin-2-one
1-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
5-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(2-hydroxyphenyl)methyl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
2-(2-methanesulfonylethyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
5-{[(propan-2-yl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amino]methyl}pyrrolidin-2-one