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2-ethyl-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)pyrimidine-5-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-ethyl-N-(oxolan-2-ylmethyl)propanamide
(1,4-dioxan-2-ylmethyl)({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-(3,4-difluorophenyl)-6-[2-(3-methylphenyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
2-amino-4-(3,5-dimethylphenyl)-6-(pyridine-2-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-[furan-2-yl(phenyl)methyl]acetamide
2-methyl-4-phenyl-9-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,9-diazaspiro[5.5]undecane
methyl (2S)-2-[3-(2-methyl-5-oxopyrrolidin-2-yl)propanamido]-3-phenylpropanoate
8-(3-ethyl-1H-pyrazole-5-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
6-(cyclopropylmethoxy)-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
3-{[1-(4-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
(4aS,8aR)-6-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
(1S,5R)-3-{[4-(benzyloxy)phenyl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{4-[(8-methoxyquinolin-2-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
4-phenyl-2-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]phenol
N,8-dimethyl-2-propyl-N-(pyrazin-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
6-(2,2-dimethylmorpholin-4-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
5-(3-methylbutyl)-5-[1-(2,3,4-trimethoxybenzoyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[(3,4-dimethoxyphenyl)methyl]-4-(piperidin-1-yl)-N-(pyridin-4-ylmethyl)benzamide
N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-[(2-fluorophenyl)methyl]-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(3-fluoro-4-methoxybenzoyl)piperidine
9-(cyclopropylmethyl)-1-methyl-4-(2-phenoxyethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(3-chloro-4-methoxyphenyl)-3-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-yl)propanamide
N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3,5-dimethoxybenzamide
1-benzyl-6-methoxy-4-[(1-methyl-1H-indol-3-yl)methyl]-1,4-diazepan-2-one
2-chloro-N-(1-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-1-phenylethyl}azepane
2-amino-4-(pyridin-3-yl)-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
6-(3,4-dimethoxybenzoyl)-1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
2-chloro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,4-dimethoxybenzamide
N-(pyridin-2-ylmethyl)-4-[5-(pyrrolidin-1-yl)pyridazin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
2-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidine-1-carbonyl)-4H-chromen-4-one
2-[5-(3-cyanophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
1-cyclohexyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-({5-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}methyl)-1,3-thiazol-2-amine
5-{1-[(2-chlorophenyl)methyl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-methyl-1H-imidazole
1-methyl-1'-(pyridine-3-sulfonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-[(3R,4S)-1-[(2,6-dimethylphenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-[2-(phenylsulfanyl)ethyl]-N-(propan-2-yl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[3-(5-methyl-4-{[(3-methylfuran-2-yl)formamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
4-(3-fluorophenoxy)-1-{[(1s,4s)-4-aminocyclohexyl]methyl}piperidine-4-carboxylic acid
2-[4-(2H-1,3-benzodioxol-5-yl)-2-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy]-N-[1-(naphthalen-1-yl)ethyl]acetamide