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N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]propanamide
2-[(4aR,7aS)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N,2-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1,3-thiazole-4-carboxamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(4-phenylazepan-1-yl)butan-1-one
6-methyl-2-(2-{4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazol-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
(3R,4S)-4-cyclopropyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-amine
5-benzenesulfonamido-1-ethyl-2-methyl-N-[3-(morpholin-4-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
2-(4-benzoylpiperazin-1-yl)-N-ethylpyridine-3-carboxamide
N-(2-hydroxy-2-phenylethyl)-N-methyl-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
N-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperidin-4-amine
3-[(1-cyclopentanecarbonylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]-N-methylbenzamide
2-methyl-4-{3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]phenyl}but-3-yn-2-ol
6-[(diethylamino)methyl]-N-[2-(1H-pyrazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(1-benzofuran-2-ylmethyl)-6-(cyclopropylmethoxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(trifluoromethyl)-1H-1,2,4-triazole
2-(hydroxymethyl)-N-(quinolin-6-yl)piperidine-1-carboxamide
4-(4-fluorophenyl)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)butanamide
5-(2-cyclopentylacetamido)-N-[(4-methoxyphenyl)methyl]-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl](1,3-thiazol-4-ylmethyl)amine
1-methyl-2-oxo-8-(quinoline-3-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-benzyl-4-(cyclopropanesulfonyl)-1-(4-methylphenyl)piperazin-2-one
N-ethyl-5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2-oxazole-3-carboxamide
3-[2-(dimethylamino)ethyl]-5-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methylphenyl)ethan-1-one
(3S,9aR)-3-[(2S)-butan-2-yl]-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-propylpyridin-2-amine
6-cyclopropyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]pyrimidin-4-amine
N-(1-{1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)acetamide
(1R,5S,6S)-6-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
2-cyclopentyl-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)-2-phenylacetamide
2-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}quinoline-4-carboxylic acid
3-[(benzyloxy)methyl]-5-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
7-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-oxa-7-azaspiro[4.5]decan-8-one
6-(2-methylpropyl)-4-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyrimidin-2-one
3-cyclopropyl-N-[2-(furan-2-yl)ethyl]-1H-pyrazole-5-carboxamide
1,2-dimethyl-3-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1H-indol-5-ol
5-(4-chloro-2-methoxyphenoxymethyl)-N-[3-(methylsulfanyl)propyl]-1,2-oxazole-3-carboxamide
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
5-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)pyridine-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(ethylamino)pyrimidine-5-carboxamide
N-(3-chloro-2-methylphenyl)-3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]propanamide
8-[(1R,2R,3S,4S)-3-aminobicyclo[2.2.1]heptane-2-carbonyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-2,2-dimethylpropan-1-ol
1-benzyl-3-[2-(2-methyl-4-phenylpiperazin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)pyrrolidine-2,5-dione
4-(methoxymethyl)-6-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidine
(3aR,5R,6S,7aS)-2-(4-butylbenzenesulfonyl)-octahydro-1H-isoindole-5,6-diol
{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}(pyridin-2-yl)methanol