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3-{2-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
9-methoxy-3-[(3-methoxyphenyl)methyl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-cyclohexyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
methyl 3-({2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazol-6-yl}formamido)propanoate
1-(2-{4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperidine
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(diphenylmethyl)-N-methyl-1,2-oxazole-5-carboxamide
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-4-yl)ethan-1-one
N-[3-(4-{[2-(3,5-difluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-3-methylbutanamide
ethyl 4-(3-{[1-2H-1,3-benzodioxol-5-yl-N-(oxolan-2-ylmethyl)formamido]methyl}-8-methylquinolin-2-yl)piperazine-1-carboxylate
7-(methylsulfanyl)-1-(pyridin-2-ylmethyl)-3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]-1,2-dihydroquinolin-2-one
9-(2-cyclopentylacetyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(methylsulfanyl)pyridine-3-carboxamide
2-amino-6-cyclobutyl-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
(1S,5R)-3-[3-(5-methylfuran-2-yl)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-methyl-1,2-oxazol-5-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
3-{1-[(2-chlorophenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
2-amino-6-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-4-ol
4-[(5-{1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
{[5-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
(3R,5S)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
2-methyl-N-(1-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
1-[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
methyl 4-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}benzoate
[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2,6-dimethylpyrimidine-4-carboxamide
N-[(2R,3R)-1'-[(2,4-dimethoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
2-(methylamino)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
N-[3-(4-hydroxyphenyl)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N,N-diethyl-1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
ethyl 1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
methyl 4-[5-({methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
1-(4-fluorophenyl)-6,6-dimethyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-(4-ethenylbenzoyl)-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-[(2E)-4-methylpent-2-en-1-yl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-{2-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl 3-benzyl-1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxylate
N'-methyl-N'-{[2-(2-methylpropoxy)phenyl]methyl}pentanediamide
6-(2,5-dimethylphenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carbonyl)morpholine
2-[(3-phenoxyazetidin-1-yl)methyl]benzonitrile
2-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]quinoxaline
(2R,3R)-3-(1H-imidazol-1-yl)-1'-(pyridin-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-phenylethyl)acetamide
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(quinolin-2-ylmethyl)amine
N-(2,2-diphenylethyl)-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
4-{[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,3-triazol-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1,3-benzothiazole
N-cyclopropyl-2-(4-fluorophenyl)-N-{[2-(4-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}acetamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide