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3-(2,3-dihydro-1H-inden-2-yl)-8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-butyl-5-(3-acetamidophenyl)furan-2-carboxamide
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N-[5-(dimethylamino)-2-methylphenyl]-4-(2-ethoxyethyl)piperazine-1-carboxamide
5-[5-(ethoxymethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-[(4-methyl-1H-imidazol-5-yl)methyl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-methanesulfonamidopropanamide
(1R,5S,6R,7S)-3-cyclopentyl-6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
[3-(2-methylpropyl)-1-(pyrimidin-2-yl)piperidin-3-yl]methanol
methyl 1-ethoxy-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[(5-methylpyrazin-2-yl)methyl]-8-(2-propoxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-N-{[8-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
1-butyl-4-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]piperidine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(methylsulfanyl)propyl]benzamide
(3R,4R)-1-[(3,5-dimethyl-1H-indol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-{1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidin-4-yl}piperidin-4-ol
2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-indole
1-(3,5-dimethylphenyl)-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperazin-2-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(pyrrolidine-1-carbonyl)piperidine
1-methyl-3-propyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
N-(1-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
6-(hydroxymethyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1,4-oxazepane-4-carboxamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[(3-methylphenyl)methyl]-1,3-oxazole-4-carboxamide
4-(2,1,3-benzoxadiazole-5-carbonyl)-1-(1H-indazol-5-yl)piperazin-2-one
1-(azocan-1-yl)-3-{4-[(benzylamino)methyl]-2-methoxyphenoxy}propan-2-ol
2-{9-[6-(1-hydroxyethyl)pyridin-2-yl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
1-[2-(4H-1,2,4-triazol-4-yl)propyl]-1H-indole
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl][(2-methyl-1H-imidazol-4-yl)methyl]amine
5-methyl-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-2-[3-(trifluoromethyl)phenyl]-1,3-oxazole
2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
1-benzyl-4-(1-benzyl-1H-pyrazole-4-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-1-(propan-2-yl)pyrrolidin-2-one
1-(4-fluorophenyl)-6,6-dimethyl-N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
(3R,5S)-N-[(2,3-difluoro-4-methoxyphenyl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-ethyl-1H-1,2,4-triazol-5-amine
2,3-dimethyl-7-[2-(3-methylphenoxy)acetyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(cyclohexylmethyl)propanamide
8-[5-(3-methoxyphenyl)furan-2-carbonyl]-1-oxa-8-azaspiro[4.5]decane
4-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(1H-imidazol-4-ylmethyl)(oxolan-2-ylmethyl)amine
4-(cyclopropylmethyl)-1-(5-ethoxyfuran-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-[2-(4-fluorophenoxymethyl)-4-hydroxypyrimidine-5-carbonyl]-2-methyl-1,4-diazepan-5-one
(3S,5S)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
3-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]-6,8-dimethyl-1,2-dihydroquinolin-2-one
(1R,5S,8R)-3-[(2,6-dichloro-3-hydroxyphenyl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methoxypiperidine
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[1-(pyridin-3-yl)propan-2-yl]propanamide
1-[(2-fluorophenyl)methyl]-N-[3-(4-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one