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1-cyclopentyl-3-(2-methoxyphenyl)-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}pyrrolidine-2,5-dione
4-(4-fluorophenyl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-4-oxobutanamide
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-(1,2-oxazinan-2-ylmethyl)phenoxy]propan-2-ol
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(5-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]azepane
3-(4-methoxyphenyl)-1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}propan-1-one
N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-4-pentanamidobenzamide
1-(3-chlorophenyl)-4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
3-[5-cyclobutyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
1-(2-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}phenyl)ethan-1-one
(3R,5S)-N-[2-(1H-imidazol-4-yl)ethyl]-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]butan-1-one
N-[4-methoxy-3-(2-methoxyacetamido)phenyl]-4-methyl-1,4-diazepane-1-carboxamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-(methoxymethyl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylcyclobutane-1-carboxamide
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
3-phenyl-N-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
3-phenyl-1-{4-[(2,4,6-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-1-ol
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
1-{2-[4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
N-(2-methoxyphenyl)-2-{3-[3-(pyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-benzyl-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carboxamide
4-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]benzonitrile
5-butyl-4-(2-methoxyacetyl)-1-(3-methylphenyl)piperazin-2-one
1-[(2,4-difluorophenyl)methyl]-5-{methyl[1-(thiophen-2-yl)ethyl]amino}azepan-2-one
N-ethyl-2-[3-(4-methoxyphenyl)-1-(3-methylbutyl)-2,5-dioxopyrrolidin-3-yl]-N-(pyridin-4-ylmethyl)acetamide
2-(2H-1,3-benzodioxol-5-yl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-[(3S,4R)-1-benzyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[(3,5-dimethoxyphenyl)methyl]propanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(5-chloropyridin-2-yl)piperazin-2-one
1-(4-chloro-2-methylphenyl)-5-[(2-methoxyethoxy)methyl]-1H-1,2,4-triazole
(cyclopropylmethyl)({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})propylamine
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]piperazin-2-one
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-methylprop-2-en-1-yl)benzamide
2-[1-(cyclohexylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N,N-diethylacetamide
2-{3-[(4-methoxyphenyl)methyl]-5-[2-(methylamino)-1,3-thiazol-4-yl]-1H-1,2,4-triazol-1-yl}acetic acid
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-methyl-8-(4-methylbenzoyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-{[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]methyl}benzonitrile
1-methyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]azepane-2-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}benzamide
3-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
2-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,3-dihydro-1,2-benzothiazol-3-one
2-(isoquinolin-1-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-(2-methylpropyl)piperidin-4-amine
2-methyl-6-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-3-yl]-3,4-dihydropyrimidin-4-one
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-[1-(1-phenylcyclopropanecarbonyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
(3R,4R)-1-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-cyclobutyl-3-methylpiperidin-4-ol