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4-(5-hydroxypyrazine-2-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}thiophene-2-carboxamide
3-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
5-ethyl-2,3-dimethyl-N-(oxolan-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}quinolin-4-ol
N-({7-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)cyclopropanecarboxamide
1-[(4-ethoxyphenyl)methyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-1H-imidazole-4-sulfonamide
methyl 4-[(2-{[benzyl({[(2S)-5-oxopyrrolidin-2-yl]methyl})amino]methyl}quinazolin-4-yl)amino]butanoate
methyl 4-{6-methoxy-4-[(4-methoxyphenyl)methyl]-3-oxo-1,4-diazepane-1-carbonyl}benzoate
2-(3-hydroxypropyl)-9-(2-methyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1,4-diazepane-1-carbonyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(4-methylpiperazine-1-carbonyl)pyrazine
4-(4-{[2-(4-methoxyphenyl)ethyl]amino}piperidin-1-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
2-phenyl-N-[2-(pyridin-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N,N-diethyl-2-{4-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
1-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
5-(3-methoxyphenoxymethyl)-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
4-{[1-cyclohexyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}phenol
(1H-imidazol-4-ylmethyl)({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
2-(2-methoxyquinolin-3-yl)pyridin-4-amine
N3,N3-diethyl-1-[(2-methoxyphenyl)methyl]-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-{[6-oxo-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-[4-(furan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-3-phenylpropan-1-ol
3-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-10-(3-hydroxypiperidine-1-carbonyl)-9-methoxy-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}propan-1-one
5-ethyl-1'-(2-methyl-1-benzofuran-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-3-ene-1-carboxamide
1-cyclohexyl-4-(5-methylthiophene-2-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
(1-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
5-benzamido-1-cyclopentyl-N-ethyl-1H-1,3-benzodiazole-7-carboxamide
3-[4-(3-propyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]-1λ6-thiolane-1,1-dione
8-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{3-[4-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-(4-oxo-4H-chromen-6-yl)piperidine-1-carboxamide
1-cyclopentanecarbonyl-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
2-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
ethyl 1-[(5-acetylthiophen-3-yl)methyl]-4-benzylpiperidine-4-carboxylate
methyl 2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-6-methylpyrimidine-4-carboxylate
1-cyclopentyl-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine
5-(3,4-difluorophenoxymethyl)-N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[3-(2-fluoro-3-methoxyphenyl)-1-methyl-1H-1,2,4-triazol-5-yl]piperidine
(3S,9aR)-3-[(benzyloxy)methyl]-8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(3-methoxyphenyl)-5-(oxan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
methyl 3-[(3,5-difluorophenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{3,5-dimethyl-4-[1-(2-methylpropyl)-5-oxopyrrolidine-3-amido]-1H-pyrazol-1-yl}acetic acid