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N-cyclopropyl-4-sulfamoyl-N-(1,3-thiazol-2-ylmethyl)benzamide
2-cyclopropyl-6-[(2S)-4-methyl-2-phenylpiperazine-1-carbonyl]-1,3-benzoxazole
N-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-(2-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N,N-dimethyl-2-[methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl})amino]propanamide
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(oxolan-3-ylmethyl)amine
N-(9H-fluoren-9-yl)-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-[2-({2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]-1,2-dihydrophthalazin-1-one
methyl 3-[(2S,4S,6R)-6-(3,5-difluorophenyl)-4-acetamidooxan-2-yl]benzoate
1-cyclohexyl-4-{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}piperazine
(2S,4R)-N,N-diethyl-4-(furan-3-amido)-1-[(3E)-pent-3-enoyl]pyrrolidine-2-carboxamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]pyridine-3-carboxamide
8-fluoro-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinoline-2-carboxamide
4-chloro-N-ethyl-2-hydroxy-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N3-(2H-1,3-benzodioxol-5-ylmethyl)-1-cyclohexyl-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
7-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decane
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[(4-methylphenyl)methyl]pyrrolidin-3-yl]methanol
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
3-[3-(1H-imidazol-1-yl)propyl]-1-[4-(morpholine-4-carbonyl)phenyl]urea
1-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
4-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
6-cyclopropyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]pyrimidin-4-amine
1-(5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
N-(furan-2-ylmethyl)-2-[2-methyl-4-oxo-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1'-[2-(pyrimidin-2-ylsulfanyl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[(2-fluorophenyl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
7-chloro-4-[2-(trifluoromethyl)morpholin-4-yl]quinoline
[5-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-4-phenyl-4H-1,2,4-triazol-3-yl]methanol
1-[(4aR,8aS)-1-(5-methylthiophene-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
N-(3-hydroxybutyl)-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
7-(cyclopropylmethyl)-2-[2-(1H-imidazol-2-yl)benzoyl]-2,7-diazaspiro[4.5]decane
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-methyl-1H-imidazole-4-carboxamide
6-(morpholine-4-carbonyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrazin-2-amine
methyl[(3-methylthiophen-2-yl)methyl]{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
(1S,6R)-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
(3aS,6aR)-5-acetyl-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-1-[2-(pyridin-3-yloxy)propyl]urea
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypyrazine
5-(1-cyclobutanecarbonylpyrrolidin-2-yl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]thiophene-2-carboxamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(piperidin-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(5-cyclohexylthiophen-2-yl)methyl]-4-(hydroxymethyl)piperidin-4-ol
2-(2,4-difluorophenoxy)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-phenylpropanamide
N-[(1S,2R)-2-aminocyclobutyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)acetamide
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-fluoro-4-methylbenzamide
1-cyclohexyl-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
1-[(2-hydroxy-6-methoxyphenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide