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2-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}benzoic acid
4-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-one
(2S,4R)-N,N-diethyl-4-(furan-3-amido)-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
1-[2-(2H-1,3-benzodioxol-5-yl)pyrimidin-4-yl]piperidin-4-ol
N,N-dimethyl-4-oxo-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butanamide
N-(furan-2-ylmethyl)-6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(oxan-4-ylmethyl)benzamide
1-(2,5-dimethoxyphenyl)-2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H-imidazole
N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-2-(naphthalen-2-yloxy)propanamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-(morpholin-3-yl)acetamide
N-(2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
3-methoxy-2-({2-methyl-2,7-diazaspiro[4.5]decan-7-yl}methyl)phenol
1-[(3,5-dimethylphenyl)methyl]-4-(3-methoxypropanoyl)piperazin-2-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-[(2-methoxyethyl)amino]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]amine
3-{[cyclohexyl(pyridin-2-ylmethyl)amino]methyl}pyrrolidin-3-ol
N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]-1,2,5-thiadiazole-3-carboxamide
2-methyl-1-{[3-(1,2-oxazinane-2-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole
2-[(3-methoxyphenyl)methyl]-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
4,6-dimethyl-2-[3-(pyridin-4-yl)azetidin-1-yl]pyridine-3-carbonitrile
3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
5-[2-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
(1S,3R)-3-amino-N-[3-(2-propoxyphenyl)propyl]cyclopentane-1-carboxamide
(2S)-2-amino-3-hydroxy-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N-methylpyridine-3-carboxamide
3-fluoro-N-(quinolin-3-ylmethyl)pyridine-4-carboxamide
1-(2-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2-dihydroquinoxalin-2-one
(1S,5R)-3-(5-methyl-1,3-benzoxazol-2-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-methylphenyl (7S,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methyl-1,3-thiazole-4-carbonyl)piperidine
2-ethyl-4-(1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)pyrimidine
4-[4-(piperidin-1-ylmethyl)benzoyl]-1λ6-thiomorpholine-1,1-dione
3-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-N-(3-hydroxyphenyl)propanamide
1-(2-{2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)-4-methyl-1H-1,2,3-triazole
5-(1H-imidazol-1-ylmethyl)-2-(4-methoxy-2,6-dimethylphenyl)pyridine
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-(quinoline-2-carbonyl)pyrrolidin-3-yl]methanol
3-(5-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
1,7-dimethyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-indole-2-carboxamide
(1S,5R)-3-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[1-(3,5-dimethylphenyl)piperidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1-[6-hydroxy-4-(5-methyl-1,3,4-thiadiazol-2-yl)-1,4-diazepan-1-yl]-3-methylbut-2-en-1-one
N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
methyl 3-{[4-(1-benzofuran-2-carbonyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
4-methyl-6-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,3-benzothiazol-2-amine
[(3R,4R)-1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-(furan-2-ylmethyl)-5-methyl-6-(4-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide