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5-(3-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-oxopropyl)-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2-methoxyquinoline-4-carboxamide
1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
N-(4-hexylphenyl)-3-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[2-(4-methylphenyl)ethyl]amino}methyl)phenoxy]propan-2-ol
6-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,6-dimethyl-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
1-[2-ethoxy-5-(trifluoromethyl)phenyl]-2-(1H-imidazol-4-yl)-1H-imidazole
(2-{4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}ethyl)dimethylamine
(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanol
(1S,5R)-3-{[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{[3-(N-methylacetamido)phenyl]methyl}acetamide
4-(2-methyl-1H-imidazol-1-yl)-N-[1-(morpholine-4-carbonyl)azepan-3-yl]butanamide
N-(furan-2-ylmethyl)-2-(methylamino)-N-(3-methylbutan-2-yl)-1,3-thiazole-4-carboxamide
[(3-chloropyridin-4-yl)methyl][(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
4-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}pyridine
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-[1-(naphthalen-1-yl)ethyl]acetamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(2,3-dihydro-1H-inden-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[4-(aminomethyl)piperidin-1-yl]-2-[(1-ethyl-1H-imidazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
3-(1H-1,2,3-benzotriazol-1-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2,3-dihydro-1-benzofuran-7-carboxamide
1-[3-oxo-3-(4-phenyl-1,4-diazepan-1-yl)propyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
N,7-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-(5-acetylthiophen-3-yl)-N-benzylacetamide
(2S)-1-(5-methyl-1,2-oxazole-3-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
(2R,3R)-3-(piperidin-1-yl)-1'-(1H-pyrazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(2S)-3-hydroxy-2-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}propanamide
6-(aminomethyl)-N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-2-methylpyrimidin-4-amine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1,3-dihydroxy-2-methylpropan-2-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(6-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}pyridin-3-yl)methyl]acetamide
2-({4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-6-methoxyphenol
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(3-fluoro-4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{4-[3-(2-methylphenyl)phenyl]-1H-1,2,3-triazol-1-yl}propanoic acid
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(1-methyl-1H-imidazole-2-carbonyl)piperidine
N-(1H-imidazol-2-ylmethyl)-N,6-dimethyl-2-propylpyrimidin-4-amine
1-{1-[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}ethan-1-one
1'-[(2-butyl-1H-imidazol-4-yl)methyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(3-chloro-4-hydroxybenzoyl)-3-ethylpiperidine-3-carboxylic acid
[(2S,4R,5R)-4-({[(4-chloro-3-fluorophenyl)methyl]amino}methyl)-5-(2-fluorophenyl)-1-methylpyrrolidin-2-yl]methanol
8-[(4-ethylphenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5-methoxy-2-{[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}-3-methyl-1H-indole
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
5-{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]pyrrolidin-2-yl}-3-methyl-1,2-oxazole
1-methanesulfonyl-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
9-[4-(4-methoxyphenyl)butanoyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
4-{methyl[(3-methyloxetan-3-yl)methyl]amino}-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide