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3-(pyridin-4-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}propanamide
3-(3-chlorobenzoyl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine
5-(oxolan-3-yl)-4-phenyl-1-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1H-imidazole
8-(2-aminopyrimidin-4-yl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(3R,5R)-1-(2-chloro-4-fluorobenzoyl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
2-(cyclopropylmethyl)-8-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
{1-[2-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]piperidin-2-yl}methanol
N-[3-(1H-imidazol-1-yl)propyl]-4-propylpyrimidine-5-carboxamide
N-({1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
2,7-dioxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-diazepane-4-carboxamide
N-[(3R,4S)-1-(furan-2-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
5-cyclopropanecarbonyl-1'-(morpholine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-4-(naphthalen-1-yl)butane-1,4-dione
(2R,6S)-4-(1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-2,6-dimethylmorpholine
2-{[2-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}carbamoyl)phenyl]amino}acetic acid
N-[(3-methoxyphenyl)methyl]-N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
1-(3-{[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]amino}propyl)pyrrolidin-2-one
3-({2-[1-(pyrrolidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[(1S,2S)-2-hydroxycyclohexyl]-3-[2-(pyridin-3-yloxy)phenyl]urea
4-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}-6-methylpyrimidin-2-amine
5-(azepane-1-sulfonyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
8-(1-tert-butyl-1H-pyrrole-3-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-(4-acetyl-1,4-diazepan-1-yl)-3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propan-1-one
2-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]propyl}-2,3-dihydro-1H-isoindol-1-one
2-[({1-[(3-chloro-4-methoxyphenyl)methyl]piperidin-3-yl}oxy)methyl]pyridine
2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
6-[(1-{[2-(dimethylamino)ethyl](methyl)amino}hex-5-en-2-yl)oxy]-N,N-dimethylpyridine-3-carboxamide
1-methyl-4-({4-methyl-5-[1-(2-methylpyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-2-(pyridin-4-yl)acetamide
1-methyl-6-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}-1H-indole
1-(thian-4-yl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]piperazine
1-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)pyrrolidin-2-one
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(2-{[(6,7-dimethyl-2-oxo-2H-chromen-4-yl)methyl]amino}ethyl)amino]-6-methyl-3,4-dihydropyrimidin-4-one
7-(cyclobutylmethyl)-2-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
8-(6-methylpyridazin-3-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[2-(2-fluorophenyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
N-(2,3-dihydro-1-benzofuran-3-yl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
5-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-2-phenylpyrimidine
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-1,7-dimethyl-1H-indole-2-carboxamide
1-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]isoquinoline
2-{[5-(1-ethoxyethyl)-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
2-cyclopropyl-4-hydroxy-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrimidine-5-carboxamide