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6-chloro-2-[(4,4-difluoropiperidin-1-yl)methyl]quinoline
2-[4-(1,3-thiazol-2-ylmethyl)piperazin-1-yl]-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazoline
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-2H-1,3-benzodioxole-5-carboxamide
2-chloro-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}benzoic acid
1-methyl-1'-{[(1s,4s)-4-aminocyclohexyl]methyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
N-(6-methoxypyridin-3-yl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}benzamide
6-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperazin-1-yl}pyrimidine-2,4-diamine
1-(5-phenyl-1,2,4-oxadiazol-3-yl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
N-(2,5-difluorophenyl)-3-[(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)amino]propanamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(pyrrolidin-1-yl)benzamide
N-(3-carbamoylphenyl)-4-[(3-methylphenyl)sulfanyl]piperidine-1-carboxamide
1-(2-methoxyacetyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-4-carboxamide
1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
4-{1-[(cyclopropylcarbamoyl)methyl]piperidin-3-yl}benzoic acid
methyl 4-{4-[2-(morpholin-2-yl)acetyl]piperazin-1-yl}benzoate
1-propyl-4-{[5-(3,3,3-trifluoropropyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(2-fluorophenyl)-N-[2-(2-methoxypyrimidine-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide
methyl 5-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-5-oxopentanoate
3-{[4-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
8-(6-aminopyridine-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(methylamino)pyridine-4-carboxamide
(3S,5R,9R)-11-(4-fluorobenzoyl)-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-(4-phenylpiperazin-1-yl)-3-[1-(3-phenylpropyl)piperidin-4-yl]propan-1-one
2-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-6-(piperidin-4-yl)-3,4-dihydropyrimidin-4-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(2-methoxypyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(5S,9aS,9bS)-5-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(6-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
1-[(ethylcarbamoyl)methyl]-4-methanesulfonyl-1,4-diazepane-6-carboxylic acid
3-{[(4-fluorophenyl)methyl]sulfanyl}-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}propan-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,5-dimethyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-({[3-hydroxy-2-oxo-1-(3-phenylpropyl)piperidin-3-yl]methyl}amino)acetamide
5-ethyl-1'-(1H-indole-6-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
1-(2-methylphenyl)-3-[1-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
N-[2-methyl-2-(morpholin-4-yl)propyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-N-(thiophen-2-ylmethyl)aniline
3-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}benzonitrile
(1-{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-yl)methanol
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-{2-[(4-chlorophenyl)methoxy]ethyl}-1-methyl-1H-pyrazole-5-carboxamide
2-(2-methoxyethyl)-9-(oxolan-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperazin-1-yl}pyrazine-2-carboxamide
N-benzyl-N-(cyclobutylmethyl)-1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane
5-{[methyl(thian-4-yl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
[(3R,4S)-1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-(3-chloro-4-methoxyphenyl)-3-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]propanamide