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2-(4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperazin-1-yl)-1,3-benzothiazole
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[4-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(2,3-dimethoxyphenyl)-3-(piperidine-1-carbonyl)pyridine
1-(2-{4-azaspiro[2.5]octan-4-ylmethyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
3-{[butyl(ethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-(2-fluorophenoxy)-1-(4-methoxypyrimidin-2-yl)piperidine-4-carboxylic acid
2-ethoxy-4-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenol
1-(3,5-dimethoxybenzoyl)-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
3-{[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}propan-1-ol
3-(dimethyl-1,2-oxazol-4-yl)-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}propanamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(3-hydroxy-2,2-dimethylpropyl)amino]methyl}piperidin-2-one
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-[2-(dimethylamino)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
5-{3-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
1-[3-(1H-imidazol-2-yl)benzoyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-benzyl-8-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
5-[1-(3,4-dimethoxyphenyl)cyclopentyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[5-methyl-2-(propan-2-yl)phenoxy]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-[1-(pyrimidin-2-yl)piperidin-3-yl]urea
4,5-dimethyl-6-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]pyrimidine
2-(4-fluorophenyl)-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
methyl[(4-methyl-1H-imidazol-5-yl)methyl]{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-{[4-(cyclopentyloxy)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
3-hydroxy-1-(3-phenylpropyl)-3-(piperidin-1-ylmethyl)piperidin-2-one
4-chloro-2-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}benzamide
3-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-[4-({methyl[(4-methylphenyl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1-{4-[hydroxy(pyridin-3-yl)methyl]piperidin-1-yl}-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-[2-(3-methoxyphenoxy)ethyl]-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-(oxan-4-yl)-6-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
5-(4-acetylphenoxymethyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
5-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-{4-[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]phenyl}-5-methyl-4H-1,2,4-triazole
2-(3-{[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]methyl}-1H-indol-1-yl)acetamide
5-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)quinoxaline
methyl 4-{4-[3-(hydroxymethyl)quinolin-2-yl]piperazin-1-yl}benzoate
2,3-dichloro-N-[(3R,5S)-5-(morpholine-4-carbonyl)pyrrolidin-3-yl]benzamide
N-[1-(1H-indol-1-yl)propan-2-yl]-5-(4-methoxyphenyl)-1,2,4-triazin-3-amine
3-cyclopropyl-5-[5-(1H-imidazol-2-yl)thiophen-2-yl]-1H-1,2,4-triazole
N-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-2-(pyridin-3-yl)piperidine-1-carboxamide
N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
5-(morpholin-4-ylmethyl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]furan-3-carboxamide
1-{3-[(butylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
3-[(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-yl)methyl]benzoic acid
2-methyl-4-[3-(pyridin-4-yl)-5-[1-(pyrrolidin-1-yl)propan-2-yl]-1H-1,2,4-triazol-1-yl]pyridine
4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one