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5-ethyl-3-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1,2,4-oxadiazole
1-(2-hydroxyethyl)-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1,4-diazepan-6-ol
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(thiophen-2-ylmethyl)acetamide
2-(2,6-dimethylpyridin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
5-methyl-3-[2-(4-methylpentyl)morpholine-4-carbonyl]-1H-indazole
3-(1-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}piperidin-3-yl)benzoic acid
[(1-cyclopentylpiperidin-4-yl)methyl][(6-methylpyridin-2-yl)methyl](pyridin-3-ylmethyl)amine
3-(hydroxymethyl)-1-(quinolin-2-ylmethyl)piperidin-3-ol
N-(3-hydroxypropyl)-1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-phenyl-4-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperazin-2-one
2-[3-(2-methoxyphenoxy)azetidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-(1H-imidazol-2-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]benzamide
2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
5-methyl-5-phenyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}piperidin-2-one
N-[(2-ethoxypyridin-3-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
ethyl 4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperazine-1-carboxylate
N-[3-(carbamoylmethyl)phenyl]-2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxylate
N-(2,2-diphenylethyl)-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[4-methyl-6-(4-{[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]amino}piperidin-1-yl)pyrimidin-2-yl]phenol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
3-benzyl-1-(1-methyl-1H-indole-3-carbonyl)piperidine-3-carboxylic acid
4-benzyl-3-ethyl-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-1,4-diazepan-5-one
3-[(dimethylamino)methyl]-1-[(2,4,6-trimethylphenyl)methyl]pyrrolidin-3-ol
1-[(3S)-3-ethylmorpholin-4-yl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
2-(2,4-difluorophenyl)-5-(2-propoxyethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,4-diazepane
({5-[1-(2,3-difluorobenzoyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-methyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-[(4-fluorophenyl)methyl]-4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-(furan-2-ylmethyl)-2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
6-methoxy-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3S,4S)-1-{[2-(furan-2-yl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
5-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
(3S,5R)-1-(2-ethylbenzoyl)-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
1-{4-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-3-(1H-pyrazol-4-yl)benzamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-(oxan-4-yl)-1H-1,3-benzodiazole-7-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)-2-(thiophen-3-yl)acetamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-fluoro-N-[(4-methoxyphenyl)methyl]benzamide
N'-(2-ethoxyphenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]propanediamide
1'-(2,3-dihydro-1-benzofuran-2-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
6-methoxy-4-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-(6-methoxypyrimidin-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-acetyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}thiophene-2-carboxamide
1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-(1,3-thiazol-4-yl)ethan-1-one