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4-[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]pyridine
1-(2-chlorophenyl)-3-{1-[1-(3-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
ethyl 2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
N-[(3S)-1-benzylpyrrolidin-3-yl]-2-propyl-1,3-thiazole-4-carboxamide
1-[(2,4,5-trimethoxyphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1-(3-methoxybenzoyl)piperidine
2-{4-[2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carbonyl]morpholin-3-yl}acetamide
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-cyclohexyl-3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]urea
3-{4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
ethyl 2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-1,3-oxazole-4-carboxylate
N-cyclooctyl-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{3-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}acetamide
4-[4-(4-methoxybutyl)piperazine-1-carbonyl]benzoic acid
3,5,7-trimethyl-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1H-indole
2-(1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidin-2-yl)acetic acid
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(5S,9aS,9bS)-5-[(E)-2-(4-fluorophenyl)ethenyl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[2-(4-fluorophenyl)azetidine-1-carbonyl]-2,6-dimethylquinoline
8-(2-aminopyrimidin-4-yl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[3-(prop-2-en-1-yl)-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-3-yl]methanol
6-[(3-hydroxypiperidin-3-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
2-[3-(piperidine-1-carbonyl)pyrazine-2-carbonyl]-2,7-diazaspiro[4.5]decane
8-{[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-2-one
5-{[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}pyrazin-2-ol
4-(8-methoxyquinolin-5-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{2-[2-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
3-cyclopentyl-1-(3-fluorophenyl)-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
2-(5-methyl-1H-pyrazol-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
N-(1-methyl-1H-indazol-3-yl)-2-[4-(9H-purin-6-yl)-1H-pyrazol-1-yl]acetamide
1-(cyclohexylmethyl)-N-ethyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-N,N-diethylpiperidine-4-carboxamide
4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1-(1,3-thiazol-2-ylmethyl)-1H-1,2,3-triazole
1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(2-methylphenoxy)piperidine-4-carboxylic acid
1-[(3-hydroxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazine
3-{2-amino-4-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methylpyrimidin-5-yl}propanoic acid
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetic acid
N-{[(2S,4S)-4-fluoro-1-(5-methylthiophene-2-carbonyl)pyrrolidin-2-yl]methyl}morpholine-4-carboxamide
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(6-oxopiperazine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,4S)-2-(2-chlorophenyl)-5-[(2,4,5-trimethoxyphenyl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
4-(2-methoxypyridin-3-yl)-N,N-dimethyl-5,6,7,8-tetrahydroquinazolin-2-amine
4-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}-N-methylbenzene-1-sulfonamide