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N-[3-(furan-2-yl)-3-phenylpropyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
3-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanoic acid
2-({2-[5-(2-methyl-1,3-thiazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)pyridine
1-({3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}methyl)-1H-pyrazole
1-[2-(dimethylamino)ethyl]-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-oxopyrrolidine-3-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(3,5-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[2-(pyridin-3-yloxy)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[2-methoxy-5-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
5-[3-(pyridin-4-yl)azetidine-1-carbonyl]quinoxaline
4-[(5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl)methyl]-1-methylpiperidine
3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-aminoethyl)-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}quinazolin-4-amine
[(2S)-1-(5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidin-2-yl]methanol
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
methyl 4-[4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]benzoate
(2S,4R)-4-amino-1-[(2-aminopyrimidin-5-yl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
(1R,5R)-6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-4-cyclopropyl-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}pyrrolidine-3-carboxylic acid
1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-3-carboxamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(pyridin-2-ylsulfanyl)acetamide
N-methyl-1-[(1s,4s)-4-aminocyclohexyl]-N-(thiophen-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-ethyl-N-methylpyridine-3-carboxamide
2-({3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
4-{4-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-{[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}-6-methyl-1,2-dihydroquinolin-2-one
2-(3-cyano-2-methyl-1H-indol-1-yl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]acetamide
2-acetyl-8-(2-hydroxynaphthalene-1-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[(4-ethoxyphenyl)methyl]-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-(thiophen-2-ylmethyl)acetamide
1-[(1S,5R)-6-(3,5-dimethyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N,N-diethyl-1-(1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-amine
1-(2-methoxy-5-{[methyl(propyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
7-(2-methoxyphenyl)-2-[3-(pyridin-2-yl)propyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-methyl-5-{4-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
4-[4-(3-fluoro-4-methylbenzoyl)-2-oxopiperazin-1-yl]benzonitrile
methyl 7-oxo-3-(1H-pyrazol-3-ylmethyl)-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-(piperidin-1-ylmethyl)-1,4-oxazepane
N-{2-[(2-chlorophenyl)formamido]ethyl}oxane-2-carboxamide
4-[2-(methylsulfanyl)pyrimidin-4-yl]-1,4-oxazepan-6-ol
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)methanesulfonamide
2-[(2,4-difluorophenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-(2-butyl-1H-imidazol-4-yl)-4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazole
[3-(2-phenoxyethyl)-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl]methanol
N,5-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazine-2-carboxamide
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-(4-phenylphenyl)ethan-1-one
(3S,4R)-4-methyl-1-(3-methyl-1-benzothiophene-2-carbonyl)piperidine-3,4-diol
5-{4-[(3-chlorophenyl)methyl]piperazine-1-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
8-[2-(2-chloro-4-methylphenoxy)ethyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N'-cyclopentyl-N-methylbutanediamide