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(2S,4R)-N-ethyl-4-{[(3-methylphenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-{[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzoic acid
6-cyclopentyl-N,1-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-methyl-4-(quinoline-2-carbonyl)piperazin-2-one
4-{4-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
N-methyl-5-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]pentanamide
N,2-dimethyl-5-(propan-2-yl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
7-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
N-[3-({[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]carbamoyl}methoxy)phenyl]propanamide
2-(3-methoxyphenyl)-N-[phenyl(pyridin-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
4-{[2-(2-aminoethyl)quinazolin-4-yl](benzyl)amino}butan-1-ol
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N3-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}piperidine-1,3-dicarboxamide
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
7-(2-hydroxyethyl)-2-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
[(3R,4R)-1-[(3-chloro-2,6-difluorophenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-5-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
3-{2-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}pyridine
[2-(4,6-dimethylpyrimidin-2-yl)ethyl]({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-(3-methylphenyl)-3-[1-(pyridine-3-sulfonyl)piperidin-4-yl]propanamide
1-(4-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethoxy}phenyl)propan-1-one
4-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}benzonitrile
1-[2-(4-chlorophenyl)propyl]-4-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazole
5-benzoyl-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(2S,4S)-4-amino-N-ethyl-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}pyrrolidine-2-carboxamide
2-(2-phenyl-1,3-thiazol-4-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-ethyl-N-(2,2,2-trifluoroethyl)acetamide
3-(thiophen-3-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propanamide
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}propan-1-one
2-[(1S,5R)-3-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
8-{[3-(2-aminoethyl)phenyl]methyl}-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2,3,6-trifluorobenzamide
1-(4-{[(1R,5S,6S)-6-(4-acetylpiperazine-1-carbonyl)-3-azabicyclo[3.1.0]hexan-3-yl]methyl}thiophen-2-yl)ethan-1-one
methyl 3-(4-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
1-(5-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-2-methoxyphenoxy)-3-(piperidin-1-yl)propan-2-ol
1-(4-chlorophenyl)-N-{[1-(4-methyl-2-oxopentanoyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
N-(2-hydroxyethyl)-N-propyl-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
9-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(1H-imidazol-2-yl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)[(1-methyl-1H-indol-5-yl)methyl]amine
N-[(4-fluorophenyl)methyl]-1-methyl-5-[4-(thiophene-2-carbonyl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N4-[(5-fluoro-2-methylphenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
1-[(4-chlorophenyl)methyl]-N-(cyclopropylmethyl)-6-oxo-N-propylpiperidine-3-carboxamide
methyl (2S)-2-{3-[(2-fluoro-5-methylphenyl)carbamoyl]propanamido}-2-phenylacetate
(4aS,8aR)-6-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(tert-butylsulfamoyl)-N-(3-fluorophenyl)-5-[(2-hydroxyethyl)amino]benzamide
(3S,4S)-4-(4-fluorophenyl)-1-(quinolin-2-ylmethyl)piperidin-3-ol
N,6-dimethyl-2-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-4-amine
5-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide