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8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2-hydroxyphenyl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
N'1-methyl-N'1-(4-methyl-1-phenylpentyl)cyclopropane-1,1-dicarboxamide
(3aS,6aS)-2-methyl-5-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
6-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-amine
5-methyl-1-(3-methylphenyl)-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-one
methyl 1-[(3R,5S)-5-{[(4-methoxyphenyl)methyl]carbamoyl}-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-ethyl-4-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine
N-[(5-methylthiophen-2-yl)methyl]-4-(2-oxopyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)butanamide
(1R,5R)-6-(5-methoxyfuran-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-(2,5-dimethoxyphenyl)-2-[4-(4-ethylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]pyrimidine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
1-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-3-(1-ethyl-1H-pyrazol-4-yl)urea
5-methoxy-1-methyl-2-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-indole
2-({5-[(4-hydroxyphenyl)methyl]-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
(1-{[1-(1-phenylpyrrolidin-3-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-2-carboxamide
1-[4-({1-ethyl-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl}methoxy)phenyl]ethan-1-one
N-(3-fluoro-4-methylphenyl)-2-{[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]amino}acetamide
(3R,4S)-4-cyclopropyl-1-(5-methylthiophene-3-carbonyl)pyrrolidin-3-amine
N-ethyl-5-(3-fluorophenoxymethyl)-N-[(1R,2R)-2-hydroxycyclohexyl]-1H-pyrazole-3-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
N-cyclopentyl-1-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
4-{6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-N-propylbenzene-1-sulfonamide
3-(2-methylphenoxy)-N-(1H-1,2,4-triazol-3-yl)azetidine-1-carboxamide
3-{[(1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2,1,3-benzothiadiazole-4-sulfonamide
N-(3-chloro-5-fluorophenyl)-3-(3-methoxypropyl)piperidine-1-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-3-(3-methyl-1H-pyrazol-1-yl)-N-(pyridin-4-ylmethyl)propanamide
(1R,5R)-6-[2-(3-chloro-4-hydroxyphenyl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-[(1H-imidazol-4-ylmethyl)amino]-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
3-ethyl-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-4-methyl-N-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(2R)-1-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)pyrrolidine-2-carboxamide
2-[1-(furan-3-ylmethyl)-4-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperazin-2-yl]ethan-1-ol
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-(4-fluorophenyl)acetamide
methyl 6-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyridine-3-carboxylate
1-(2-phenylphenyl)-4-[2-(1H-1,2,4-triazol-1-yl)propanoyl]piperazin-2-one
methyl 2-(3-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}-1H-indol-1-yl)acetate
5-(2,4-difluorophenoxymethyl)-N-[(1r,4r)-4-hydroxycyclohexyl]-1,2-oxazole-3-carboxamide
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]acetamide
5-methyl-N-[(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-3-yl)methyl]pyrazine-2-carboxamide
({3-[2-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-2-yl)ethoxy]phenyl}methyl)(methyl)(quinolin-8-ylmethyl)amine
4-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one
4-[2-(4-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}phenoxy)ethyl]morpholine
(3aR,5R,6S,7aS)-2-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-octahydro-1H-isoindole-5,6-diol
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(3-methoxyphenyl)acetamide
2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-(thiophen-3-yl)acetic acid
(3S,9aR)-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2,3-dimethyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione