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1-(2-methoxy-4-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
1-(3-{4-[(cyclooctylamino)methyl]-2-methoxyphenoxy}-2-hydroxypropyl)piperidin-4-ol
methyl 2-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonyl}-6-[(3,4-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[3-chloro-5-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
1-methyl-N-{2-[methyl(phenyl)amino]ethyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-(5-methylthiophen-2-yl)-N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-1H-pyrazole-5-carboxamide
3-{[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
N-[(4-phenyloxan-4-yl)methyl]-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
ethyl 3-benzyl-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine-3-carboxylate
4-{4-[4-(pyrrolidin-1-yl)piperidin-1-yl]pyridine-2-carbonyl}morpholine
5-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]-2-(methoxymethyl)pyrimidine
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,5-dimethylfuran-2-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[3-(3-methoxyphenoxy)azetidin-1-yl]ethan-1-one
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]propanamide
1-(2,3-dihydro-1H-indol-1-yl)-2-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-3-(2-oxopyrrolidin-1-yl)propanamide
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-(phenylamino)pyrimidine-5-carboxamide
N-(4-ethenylphenyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
N-(3-{2-methoxy-4-[(3-methylpiperidin-1-yl)methyl]phenoxy}propyl)-4-(trifluoromethyl)benzamide
N-(3,3-diphenylpropyl)-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
4-({2-[1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(pyrrolidine-1-sulfonyl)ethyl]amine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-{3-[2-(2-fluoro-4,5-dimethoxyphenyl)-1H-imidazol-1-yl]propyl}morpholine
(3R,5R)-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
(4aS,8aR)-6-(2-hydroxyacetyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-3-[4-({[(1-hydroxycyclohexyl)methyl]carbamoyl}amino)phenyl]propanamide
7-fluoro-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}quinazolin-4-amine
N-(1,3-dihydro-2-benzofuran-5-yl)-1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-carboxamide
2-methoxy-5-{[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}benzoic acid
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(4-methylphenoxy)ethan-1-one
2-[(4-methoxyphenyl)methyl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}morpholine
8-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,8aR)-6-(2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-methoxy-1-{[2-(methylsulfanyl)phenyl]methyl}piperidine
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-(quinoxalin-2-ylmethyl)benzamide
2-[5-(3,4-dimethylphenoxymethyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
{[(1R,5S,6R)-3-cyclopropanecarbonyl-3-azabicyclo[3.1.0]hexan-6-yl]methyl}[(4-methylphenyl)methyl](prop-2-yn-1-yl)amine
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
{4-[(4-methoxyphenyl)methyl]-1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl}methanol
2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyridine-4-carboxamide
(3R,4R)-1-[2-(dimethylamino)pyridine-3-carbonyl]-3,4-dimethylpyrrolidin-3-ol
N-ethyl-2-(1H-imidazol-2-yl)-N-(pyridin-4-ylmethyl)benzamide
N-methyl-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(4-methylphenoxy)ethyl]propanamide
3-{[(1,3-dihydroxypropan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-[4-(benzyloxy)-2-hydroxyphenyl]-1,3-dimethyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[(2-methylphenyl)methyl]-4-(oxane-4-carbonyl)piperazine