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4-oxo-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(1R,7S)-3-[(4-fluorophenyl)methyl]-6-(3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-{[4-(2-hydroxyethoxy)phenyl]methyl}-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
(3R,4R)-4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1-(4-methoxybenzoyl)pyrrolidin-3-ol
3-[1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]aniline
9-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
1-[3-(methylsulfanyl)propyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N3-[(2,6-difluoro-3-methylphenyl)methyl]-N5-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(dicyclopropylmethyl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
6-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2-acetamido-3-methylbutanamide
(4aS,8aR)-2-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)-decahydroisoquinoline
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(morpholin-4-yl)propan-1-one
(2S)-1-acetyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
1-(1,2,5-oxadiazole-3-carbonyl)-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
2-(5-methyl-1,2-oxazol-3-yl)-1-[4-(piperidin-1-ylmethyl)benzoyl]piperidine
N-[3-({[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]carbamoyl}amino)-4-fluorophenyl]acetamide
5-ethyl-N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[methyl(pyridin-2-ylmethyl)amino]acetamide
N-(2-hydroxyethyl)-2-(phenylamino)-N-(1,3-thiazol-2-ylmethyl)pyrimidine-5-carboxamide
2-benzyl-8-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)propanamide
4-(1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)morpholine
(2E)-N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-3-(thiophen-2-yl)prop-2-enamide
4-methyl-2-({4-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)phenol
N-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
2-{2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(1,3,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-ol
N-(4-hydroxybutyl)-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamide
1-[(5-chlorothiophen-2-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
1-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-4-oxo-1,4-dihydroquinoline-3-carboxamide
3-[1-(2,6-dimethoxypyrimidine-4-carbonyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
5-(3-methylphenyl)-4-[1-(oxolane-2-carbonyl)piperidin-4-yl]-2-(pyridin-4-yl)pyrimidine
(2S,4S)-4-amino-N-ethyl-1-(3-methylfuran-2-carbonyl)pyrrolidine-2-carboxamide
6-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,7S)-N-(2-hydroxyethyl)-N-methyl-4-oxo-3-[2-(piperidin-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-[(dimethylamino)methyl]-N-(5-fluoro-2-methylphenyl)-4-hydroxyazepane-1-carboxamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N'-(3-chloro-2-methylphenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]propanediamide
2-(4-methyl-1H-pyrazol-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]propanamide
N-(1,3-benzoxazol-2-ylmethyl)-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
(2S)-N-[2-(2,4-dimethylphenoxy)ethyl]-2-hydroxy-N-methylpropanamide
1-(furan-3-carbonyl)-4-(2-methoxyphenoxy)piperidine
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-N-[2-(1H-imidazol-4-yl)ethyl]-5-[(pyridin-3-yloxy)methyl]piperidine-3-carboxamide
N-{4-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-amine
6-(4-hydroxypiperidin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
4-{3-[4-(2-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[(4-methyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[3-(dimethylamino)propyl]-1-benzothiophene-5-carboxamide