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N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carboxamide
(1S,5R)-6-(3-chloro-4-methylbenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)piperazin-1-yl]-1-(piperidin-1-yl)ethan-1-one
2-methyl-6-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)pyrrolidine-1-carboxamide
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-4-(propan-2-yl)pyrimidin-2-amine
1-(2-chlorophenyl)-4-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine
8-[(4-methoxypyridin-2-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
4-{3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-cyclohexyl-2-(2-oxopiperidin-1-yl)-N-(thiophen-3-ylmethyl)acetamide
4-{2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-1λ6-thiane-1,1-dione
({4-[1-(2,3-dihydro-1H-inden-2-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-yl}methyl)dimethylamine
ethyl({[2-(furan-2-yl)pyrimidin-5-yl]methyl})(oxan-4-ylmethyl)amine
6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N-(propan-2-yl)pyridazin-3-amine
1-{2-[methyl({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})amino]ethyl}cyclopentan-1-ol
(3S,4R)-N,N-dimethyl-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-amine
1-{4-[(pentan-3-yl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
methyl 1-{1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carbonyl}piperidine-2-carboxylate
N-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]thiomorpholine-4-carboxamide
2-[3-(3,4-difluorophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
(1H-1,3-benzodiazol-2-ylmethyl)(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
ethyl 1-{2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetyl}piperidine-2-carboxylate
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-[1-(pyrazin-2-yl)piperidin-3-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-methyl-N-(4-{1-[(methylcarbamoyl)methyl]-1H-pyrazol-4-yl}phenyl)propanamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
2-methyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrido[2,3-d]pyrimidin-4-amine
4-(4-chloro-3-fluorobenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-[2-(cyclohex-1-ene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
1-(7-fluoro-2-methylquinoline-4-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
4-{1-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
(2S,3R)-3-hydroxy-2-{[2-(4-methoxyphenoxymethyl)-1,3-oxazol-4-yl]formamido}butanamide
(4aS,8aR)-6-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-1-butyl-decahydro-1,6-naphthyridin-2-one
3-[(dimethylamino)methyl]-1-(3-hydroxy-4-methoxybenzoyl)pyrrolidin-3-ol
4-(3-methylfuran-2-carbonyl)-1,4-diazepan-2-one
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methylphenyl)methyl]piperidine
1-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-3-phenylprop-2-yn-1-one
4-hydroxy-1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidine-4-carboxylic acid
3-(2,5-dioxoimidazolidin-4-yl)-N-[(2-propyl-1,3-thiazol-4-yl)methyl]propanamide
N-benzyl-5-(4-cyclopentylpiperazine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
7-[4-(1H-pyrazol-1-yl)benzoyl]-1-oxa-7-azaspiro[3.5]nonane
2-{1-azabicyclo[3.2.1]octan-5-yloxy}-6-fluorobenzonitrile
3-(4-benzyl-1H-pyrazol-5-yl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
4,6-dimethyl-3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
3-butanamido-N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]benzamide
8-[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[3-(2-methyl-1H-imidazol-1-yl)propyl]amine
2-(3-hydroxypropyl)-9-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-1-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(quinolin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one